XMD8-92 KiNativ -- single dose experiment - Dataset - HMS LINCS Database

XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small molecules	Cells	Proteins

Small Molecule	Cell Line	Protein	Sequence	Labeling Site	% Inhibition	Assay compound conc	Conc unit
XMD8-92	HeLa	CDK2	DLkPQNLLINTEGAIK	Lys2	-18.6	10	uM
XMD8-92	PC-3	CDK2	DLkPQNLLINTEGAIK	Lys2	9.2	10	uM
XMD8-92	PC-3	CDK5	DLkPQNLLINR	Lys2	-1.0	10	uM
XMD8-92	PC-3	CDK5	NRETHEIVALkR	Lys1	1.0	10	uM
XMD8-92	PC-3	CDK5	ETHEIVALkR	Lys1	-8.6	10	uM
XMD8-92	HeLa	CDK7	DLkPNNLLLDENGVLK	Lys2	-11.2	10	uM
XMD8-92	PC-3	CDK9	DMkAANVLITR	Lys2	-16.1	10	uM
XMD8-92	HeLa	CHK1	DIkPENLLLDER	Lys2	1.3	10	uM
XMD8-92	PC-3	CHK2	VAIkIISK	Lys1	2.6	10	uM
XMD8-92	PC-3	CHK2	DLkPENVLLSSQEEDCLIK	Lys2	8.3	10	uM
XMD8-92	HeLa	CHK2	DLkPENVLLSSQEEDCLIK	Lys2	-1.4	10	uM
XMD8-92	PC-3	CK1d,CK1e	DVkPDNFLMGLGKK	Lys2	-5.8	10	uM
XMD8-92	PC-3	CLK2	LTHTDLkPENILFVNSDYELTYNLEK	Lys2	-15.6	10	uM
XMD8-92	HeLa	CSK	VSDFGLTkEASSTQDTGKLPVK	Activation Loop	-7.0	10	uM
XMD8-92	PC-3	CSK	VSDFGLTkEASSTQDTGKLPVK	Activation Loop	-16.1	10	uM
XMD8-92	HeLa	DGKA	IDPVPNTHPLLVFVNPkSGGK	ATP	-25.7	10	uM
XMD8-92	HeLa	DMPK	DIkPDNILLDR	Lys2	-15.7	10	uM
XMD8-92	PC-3	DNAPK	GHDEREHPFLVkGGEDLRQDQR	ATP	0.1	10	uM
XMD8-92	HeLa	DNAPK	GHDEREHPFLVkGGEDLRQDQR	ATP	-7.2	10	uM
XMD8-92	PC-3	DNAPK	kGGSWIQEINVAEK	ATP	11.8	10	uM
XMD8-92	PC-3	eEF2K	YIkYNSNSGFVR	Protein Kinase Domain	-5.5	10	uM
XMD8-92	HeLa	eEF2K	YIkYNSNSGFVR	Protein Kinase Domain	-13.5	10	uM
XMD8-92	PC-3	EGFR	ITDFGLAkLLGAEEK	Activation Loop	-4.3	10	uM
XMD8-92	PC-3	EGFR	LLGAEEKEYHAEGGkVPIK	Activation Loop	-3.2	10	uM
XMD8-92	PC-3	EGFR	IPVAIkELR	Lys1	-5.4	10	uM