XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-50.1
10
uM
XMD8-92 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
6.9
10
uM
XMD8-92 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
3.4
10
uM
XMD8-92 HeLa TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD8-92 PC-3 TLK1
YAAVkIHQLNK
Lys1
13.2
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-12.6
10
uM
XMD8-92 HeLa ULK3
EVVAIkCVAK
Lys1
1.6
10
uM
XMD8-92 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-6.2
10
uM
XMD8-92 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-10.4
10
uM
XMD8-92 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-1.9
10
uM
XMD8-92 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
8.8
10
uM
XMD8-92 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-24.3
10
uM
XMD8-92 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
0.5
10
uM