XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-7.3
10
uM
XMD8-92 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
7.3
10
uM
XMD8-92 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
10
uM
XMD8-92 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
7.3
10
uM
XMD8-92 PC-3 KHS1
NVHTGELAAVkIIK
Lys1
-7.6
10
uM
XMD8-92 HeLa PKD2
DVAVkVIDK
Lys1
7.6
10
uM
XMD8-92 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.6
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
7.9
10
uM
XMD8-92 PC-3 CDK10
DLkVSNLLMTDK
Lys2
-8.1
10
uM
XMD8-92 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-8.3
10
uM
XMD8-92 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
8.3
10
uM
XMD8-92 HeLa MAP2K3
DVkPSNVLINK
Lys2
8.3
10
uM
XMD8-92 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-8.6
10
uM
XMD8-92 PC-3 CDK5
ETHEIVALkR
Lys1
-8.6
10
uM
XMD8-92 HeLa SGK3
FYAVkVLQK
Lys1
-8.8
10
uM
XMD8-92 PC-3 MK11
QELNkTVWEVPQR
Other
8.8
10
uM
XMD8-92 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
8.8
10
uM
XMD8-92 HeLa MASTL
LYAVkVVK
Lys1
8.9
10
uM
XMD8-92 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
8.9
10
uM
XMD8-92 HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
9.0
10
uM
XMD8-92 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
9.1
10
uM
XMD8-92 HeLa MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
9.1
10
uM
XMD8-92 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-9.2
10
uM
XMD8-92 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-9.2
10
uM