XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -7.3 | 10 | uM |
XMD8-92 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | 7.3 | 10 | uM |
XMD8-92 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 7.3 | 10 | uM |
XMD8-92 | HeLa | IRAK3 | SHLEHQSCTINMTSSSSkHLWYMPEEYIR | Protein Kinase Domain | 7.3 | 10 | uM |
XMD8-92 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | -7.6 | 10 | uM |
XMD8-92 | HeLa | PKD2 | DVAVkVIDK | Lys1 | 7.6 | 10 | uM |
XMD8-92 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 7.6 | 10 | uM |
XMD8-92 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 7.8 | 10 | uM |
XMD8-92 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 7.9 | 10 | uM |
XMD8-92 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | -8.1 | 10 | uM |
XMD8-92 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.3 | 10 | uM |
XMD8-92 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -8.6 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -8.6 | 10 | uM |
XMD8-92 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |
XMD8-92 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 8.8 | 10 | uM |
XMD8-92 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 8.8 | 10 | uM |
XMD8-92 | HeLa | MASTL | LYAVkVVK | Lys1 | 8.9 | 10 | uM |
XMD8-92 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 8.9 | 10 | uM |
XMD8-92 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 9.0 | 10 | uM |
XMD8-92 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 9.1 | 10 | uM |
XMD8-92 | HeLa | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | 9.1 | 10 | uM |
XMD8-92 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -9.2 | 10 | uM |
XMD8-92 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | -9.2 | 10 | uM |