XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -1.4 | 10 | uM |
| XMD8-92 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -1.4 | 10 | uM |
| XMD8-92 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | 14.2 | 10 | uM |
| XMD8-92 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 1.5 | 10 | uM |
| XMD8-92 | PC-3 | MAP2K3 | DVkPSNVLINK | Lys2 | 1.5 | 10 | uM |
| XMD8-92 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 15.0 | 10 | uM |
| XMD8-92 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 15.1 | 10 | uM |
| XMD8-92 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | -15.2 | 10 | uM |
| XMD8-92 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -15.5 | 10 | uM |
| XMD8-92 | PC-3 | CLK2 | LTHTDLkPENILFVNSDYELTYNLEK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 15.6 | 10 | uM |
| XMD8-92 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -15.7 | 10 | uM |
| XMD8-92 | HeLa | PIK3CG | KkPLWLEFK | ATP | -15.8 | 10 | uM |
| XMD8-92 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -15.9 | 10 | uM |
| XMD8-92 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | -1.6 | 10 | uM |
| XMD8-92 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 1.6 | 10 | uM |
| XMD8-92 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 1.6 | 10 | uM |
| XMD8-92 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | 1.6 | 10 | uM |
| XMD8-92 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -16.1 | 10 | uM |
| XMD8-92 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | -16.1 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
| XMD8-92 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -1.7 | 10 | uM |
| XMD8-92 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | 17.4 | 10 | uM |
| XMD8-92 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 17.5 | 10 | uM |