XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 10.9 | 10 | uM |
XMD8-92 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -11.0 | 10 | uM |
XMD8-92 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 11.1 | 10 | uM |
XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -11.4 | 10 | uM |
XMD8-92 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -11.5 | 10 | uM |
XMD8-92 | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | -11.5 | 10 | uM |
XMD8-92 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -11.6 | 10 | uM |
XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
XMD8-92 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 11.8 | 10 | uM |
XMD8-92 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -11.9 | 10 | uM |
XMD8-92 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -12.5 | 10 | uM |
XMD8-92 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 12.5 | 10 | uM |
XMD8-92 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -12.6 | 10 | uM |
XMD8-92 | PC-3 | PKCa,PKCb | DLkLDNVMLDSEGHIK | Lys2 | -12.7 | 10 | uM |
XMD8-92 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -1.3 | 10 | uM |
XMD8-92 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | 1.3 | 10 | uM |
XMD8-92 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 1.3 | 10 | uM |
XMD8-92 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -13.0 | 10 | uM |
XMD8-92 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -13.2 | 10 | uM |
XMD8-92 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | 13.2 | 10 | uM |
XMD8-92 | PC-3 | MK14 | QELNkTIWEVPER | Other | 13.3 | 10 | uM |
XMD8-92 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.5 | 10 | uM |
XMD8-92 | HeLa | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 13.6 | 10 | uM |