XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
10.9
10
uM
XMD8-92 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-11.0
10
uM
XMD8-92 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
11.1
10
uM
XMD8-92 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-11.2
10
uM
XMD8-92 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-11.2
10
uM
XMD8-92 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
-11.4
10
uM
XMD8-92 HeLa LATS2
VDTHALYAMkTLR
Lys1
-11.5
10
uM
XMD8-92 HeLa PKR
DLkPSNIFLVDTK
Lys2
-11.5
10
uM
XMD8-92 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-11.6
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
11.7
10
uM
XMD8-92 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
11.8
10
uM
XMD8-92 HeLa NEK9
LGDYGLAkK
Activation Loop
-11.9
10
uM
XMD8-92 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-12.5
10
uM
XMD8-92 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
12.5
10
uM
XMD8-92 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-12.6
10
uM
XMD8-92 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
-12.7
10
uM
XMD8-92 HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
-1.3
10
uM
XMD8-92 HeLa CHK1
DIkPENLLLDER
Lys2
1.3
10
uM
XMD8-92 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
1.3
10
uM
XMD8-92 HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-13.0
10
uM
XMD8-92 HeLa KS6B2
DLkPENIMLSSQGHIK
Lys2
-13.2
10
uM
XMD8-92 PC-3 TLK1
YAAVkIHQLNK
Lys1
13.2
10
uM
XMD8-92 PC-3 MK14
QELNkTIWEVPER
Other
13.3
10
uM
XMD8-92 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.5
10
uM
XMD8-92 HeLa MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
13.6
10
uM