XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa BTK
GQYDVAIkMIK
Lys1
-9.2
10
uM
XMD8-92 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
9.2
10
uM
XMD8-92 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
9.2
10
uM
XMD8-92 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
-9.3
10
uM
XMD8-92 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-9.3
10
uM
XMD8-92 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
9.3
10
uM
XMD8-92 PC-3 PI42C
ELPTLkDMDFLNK
ATP
9.3
10
uM
XMD8-92 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
-9.4
10
uM
XMD8-92 PC-3 GCN2
LDGCCYAVkR
Lys1
9.4
10
uM
XMD8-92 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.0
10
uM
XMD8-92 HeLa LOK
NKETGALAAAkVIETK
Lys1
-9.7
10
uM
XMD8-92 HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
-9.7
10
uM
XMD8-92 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
9.7
10
uM
XMD8-92 HeLa AurB
SHFIVALkVLFK
Lys1
9.7
10
uM