XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 8.8 | 10 | uM |
| XMD8-92 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -24.3 | 10 | uM |
| XMD8-92 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 0.5 | 10 | uM |
| XMD8-92 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 9.3 | 10 | uM |
| XMD8-92 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | -1.0 | 10 | uM |
| XMD8-92 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | 1.3 | 10 | uM |
| XMD8-92 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -1.4 | 10 | uM |
| XMD8-92 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 8.3 | 10 | uM |
| XMD8-92 | HeLa | MYO3A,MYO3B | DVkGNNILLTTEGGVK | Lys2 | -19.5 | 10 | uM |
| XMD8-92 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -9.7 | 10 | uM |
| XMD8-92 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -35.4 | 10 | uM |
| XMD8-92 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -3.9 | 10 | uM |
| XMD8-92 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -12.6 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
| XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
| XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -15.5 | 10 | uM |
| XMD8-92 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | -8.1 | 10 | uM |
| XMD8-92 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 2.8 | 10 | uM |
| XMD8-92 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -18.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 9.2 | 10 | uM |
| XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
| XMD8-92 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | -16.1 | 10 | uM |
| XMD8-92 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -1.7 | 10 | uM |
| XMD8-92 | PC-3 | MK14 | QELNkTIWEVPER | Other | 13.3 | 10 | uM |