XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -3.6 | 10 | uM |
XMD8-92 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -18.1 | 10 | uM |
XMD8-92 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 3.9 | 10 | uM |
XMD8-92 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 7.2 | 10 | uM |
XMD8-92 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | -0.8 | 10 | uM |
XMD8-92 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 10.9 | 10 | uM |
XMD8-92 | PC-3 | CDK14 | LVALkVIR | Lys1 | -6.6 | 10 | uM |
XMD8-92 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | -43.4 | 10 | uM |
XMD8-92 | PC-3 | ILK | WQGNDIVVkVLK | Lys1 | 17.7 | 10 | uM |
XMD8-92 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 1.6 | 10 | uM |
XMD8-92 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 2.7 | 10 | uM |
XMD8-92 | HeLa | LATS1 | ALYATkTLR | Lys1 | 0.4 | 10 | uM |
XMD8-92 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 7.8 | 10 | uM |
XMD8-92 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.9 | 10 | uM |
XMD8-92 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -6.3 | 10 | uM |
XMD8-92 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 17.5 | 10 | uM |
XMD8-92 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 6.7 | 10 | uM |
XMD8-92 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | 1.8 | 10 | uM |
XMD8-92 | PC-3 | CHK2 | VAIkIISK | Lys1 | 2.6 | 10 | uM |
XMD8-92 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 40.4 | 10 | uM |
XMD8-92 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -26.2 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 1.0 | 10 | uM |
XMD8-92 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 5.2 | 10 | uM |
XMD8-92 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -2.2 | 10 | uM |
XMD8-92 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |