XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa CAMK1D
LFAVkCIPK
Lys1
-3.6
10
uM
XMD8-92 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-18.1
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
3.9
10
uM
XMD8-92 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
7.2
10
uM
XMD8-92 HeLa MLTK
WISQDKEVAVKk
Lys1
-0.8
10
uM
XMD8-92 PC-3 MLTK
WISQDKEVAVKk
Lys1
10.9
10
uM
XMD8-92 PC-3 CDK14
LVALkVIR
Lys1
-6.6
10
uM
XMD8-92 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
-43.4
10
uM
XMD8-92 PC-3 ILK
WQGNDIVVkVLK
Lys1
17.7
10
uM
XMD8-92 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
1.6
10
uM
XMD8-92 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
2.7
10
uM
XMD8-92 HeLa LATS1
ALYATkTLR
Lys1
0.4
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 HeLa ILK
WQGNDIVVkVLK
Lys1
-4.9
10
uM
XMD8-92 HeLa CaMK1a
LVAIkCIAK
Lys1
-6.3
10
uM
XMD8-92 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
17.5
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
6.7
10
uM
XMD8-92 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
1.8
10
uM
XMD8-92 PC-3 CHK2
VAIkIISK
Lys1
2.6
10
uM
XMD8-92 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
40.4
10
uM
XMD8-92 HeLa GCK
DTVTSELAAVkIVK
Lys1
-26.2
10
uM
XMD8-92 PC-3 CDK5
NRETHEIVALkR
Lys1
1.0
10
uM
XMD8-92 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
5.2
10
uM
XMD8-92 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
-2.2
10
uM
XMD8-92 HeLa SGK3
FYAVkVLQK
Lys1
-8.8
10
uM