XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa MK14
QELNkTIWEVPER
Other
4.1
10
uM
XMD8-92 PC-3 MK11
QELNkTVWEVPQR
Other
8.8
10
uM
XMD8-92 PC-3 ROCK1
kLQLELNQER
Other
-4.3
10
uM
XMD8-92 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-10.4
10
uM
XMD8-92 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
10
uM
XMD8-92 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
22.4
10
uM
XMD8-92 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.5
10
uM
XMD8-92 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-9.2
10
uM
XMD8-92 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
6.0
10
uM
XMD8-92 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
7.3
10
uM
XMD8-92 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
2.6
10
uM
XMD8-92 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-20.2
10
uM
XMD8-92 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-5.5
10
uM
XMD8-92 HeLa PAN3
VMDPTkILITGK
-4.5
10
uM