XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 6.6 | 10 | uM |
XMD8-92 | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | -17.9 | 10 | uM |
XMD8-92 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 1.6 | 10 | uM |
XMD8-92 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -3.2 | 10 | uM |
XMD8-92 | HeLa | KPCI | IYAMkVVK | Lys1 | 4.3 | 10 | uM |
XMD8-92 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | 0.9 | 10 | uM |
XMD8-92 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 10.0 | 10 | uM |
XMD8-92 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 18.5 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -8.6 | 10 | uM |
XMD8-92 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -4.3 | 10 | uM |
XMD8-92 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -9.2 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -10.5 | 10 | uM |
XMD8-92 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -5.7 | 10 | uM |
XMD8-92 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 10.7 | 10 | uM |
XMD8-92 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -5.2 | 10 | uM |
XMD8-92 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 9.4 | 10 | uM |
XMD8-92 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -9.3 | 10 | uM |
XMD8-92 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -68.4 | 10 | uM |
XMD8-92 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 3.9 | 10 | uM |
XMD8-92 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | -4.6 | 10 | uM |
XMD8-92 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | -20.9 | 10 | uM |
XMD8-92 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 8.8 | 10 | uM |
XMD8-92 | PC-3 | PDK1 | EYAIkILEK | Lys1 | 4.9 | 10 | uM |
XMD8-92 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 9.3 | 10 | uM |
XMD8-92 | HeLa | PKD2 | DVAVkVIDK | Lys1 | 7.6 | 10 | uM |