XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-7.0
10
uM
XMD8-92 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
4.2
10
uM
XMD8-92 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
2.8
10
uM
XMD8-92 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
2.7
10
uM
XMD8-92 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
-10.9
10
uM
XMD8-92 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-10.4
10
uM
XMD8-92 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-18.1
10
uM
XMD8-92 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
6.5
10
uM
XMD8-92 HeLa JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-0.1
10
uM
XMD8-92 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
-7.2
10
uM
XMD8-92 HeLa SGK3
FYAVkVLQK
Lys1
-8.8
10
uM
XMD8-92 HeLa LATS1
ALYATkTLR
Lys1
0.4
10
uM
XMD8-92 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-8.3
10
uM
XMD8-92 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.5
10
uM
XMD8-92 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
15.0
10
uM
XMD8-92 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-15.6
10
uM
XMD8-92 HeLa LOK
NKETGALAAAkVIETK
Lys1
-9.7
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-16.3
10
uM
XMD8-92 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-11.6
10
uM
XMD8-92 HeLa MAP3K5,MAP3K6,MAP3K7
IAIkEIPERDSR
Lys1
3.2
10
uM
XMD8-92 HeLa MAP2K3
DVkPSNVLINK
Lys2
8.3
10
uM
XMD8-92 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-20.3
10
uM
XMD8-92 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
-18.6
10
uM
XMD8-92 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
-43.4
10
uM
XMD8-92 HeLa MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
18.1
10
uM