XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -7.0 | 10 | uM |
XMD8-92 | HeLa | PKD1,PKD2 | NIVHCDLkPENVLLASADPFPQVK | Lys2 | 4.2 | 10 | uM |
XMD8-92 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 2.8 | 10 | uM |
XMD8-92 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 2.7 | 10 | uM |
XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
XMD8-92 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | -10.4 | 10 | uM |
XMD8-92 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -18.1 | 10 | uM |
XMD8-92 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | 6.5 | 10 | uM |
XMD8-92 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -0.1 | 10 | uM |
XMD8-92 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -7.2 | 10 | uM |
XMD8-92 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |
XMD8-92 | HeLa | LATS1 | ALYATkTLR | Lys1 | 0.4 | 10 | uM |
XMD8-92 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.3 | 10 | uM |
XMD8-92 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.5 | 10 | uM |
XMD8-92 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 15.0 | 10 | uM |
XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
XMD8-92 | HeLa | LOK | NKETGALAAAkVIETK | Lys1 | -9.7 | 10 | uM |
XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
XMD8-92 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -11.6 | 10 | uM |
XMD8-92 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | 3.2 | 10 | uM |
XMD8-92 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -20.3 | 10 | uM |
XMD8-92 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -18.6 | 10 | uM |
XMD8-92 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | -43.4 | 10 | uM |
XMD8-92 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 18.1 | 10 | uM |