XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
8.3
10
uM
XMD8-92 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
10.0
10
uM
XMD8-92 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
9.1
10
uM
XMD8-92 PC-3 NEK8
DLkTQNILLDK
Lys2
4.0
10
uM
XMD8-92 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-3.7
10
uM
XMD8-92 PC-3 NEK9
DIkTLNIFLTK
Lys2
5.6
10
uM
XMD8-92 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
18.5
10
uM
XMD8-92 PC-3 NEK9
LGDYGLAkK
Activation Loop
5.0
10
uM
XMD8-92 PC-3 CDK5
ETHEIVALkR
Lys1
-8.6
10
uM
XMD8-92 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
6.1
10
uM
XMD8-92 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-4.3
10
uM
XMD8-92 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
4.6
10
uM
XMD8-92 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-7.3
10
uM
XMD8-92 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-9.2
10
uM