XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
6.6
10
uM
XMD8-92 PC-3 SRPK1/2
FVAMkVVK
Lys1
-17.9
10
uM
XMD8-92 HeLa ULK3
EVVAIkCVAK
Lys1
1.6
10
uM
XMD8-92 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-3.2
10
uM
XMD8-92 HeLa KPCI
IYAMkVVK
Lys1
4.3
10
uM
XMD8-92 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
0.9
10
uM
XMD8-92 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
10.0
10
uM
XMD8-92 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
18.5
10
uM
XMD8-92 PC-3 CDK5
ETHEIVALkR
Lys1
-8.6
10
uM
XMD8-92 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-4.3
10
uM
XMD8-92 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-9.2
10
uM
XMD8-92 PC-3 EPHA2
EVPVAIkTLK
Lys1
-10.5
10
uM
XMD8-92 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-5.7
10
uM
XMD8-92 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
10.7
10
uM
XMD8-92 HeLa GCN2
LDGCCYAVkR
Lys1
-5.2
10
uM
XMD8-92 PC-3 GCN2
LDGCCYAVkR
Lys1
9.4
10
uM
XMD8-92 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-9.3
10
uM
XMD8-92 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-68.4
10
uM
XMD8-92 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
3.9
10
uM
XMD8-92 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
-4.6
10
uM
XMD8-92 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
-20.9
10
uM
XMD8-92 PC-3 MK11
QELNkTVWEVPQR
Other
8.8
10
uM
XMD8-92 PC-3 PDK1
EYAIkILEK
Lys1
4.9
10
uM
XMD8-92 PC-3 PI42C
ELPTLkDMDFLNK
ATP
9.3
10
uM
XMD8-92 HeLa PKD2
DVAVkVIDK
Lys1
7.6
10
uM