XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
-15.5
10
uM
XMD8-92 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
9.3
10
uM
XMD8-92 HeLa AurB
SHFIVALkVLFK
Lys1
9.7
10
uM
XMD8-92 HeLa ATR
FYIMMCkPK
ATP
-5.7
10
uM
XMD8-92 PC-3 ATR
FYIMMCkPK
ATP
6.1
10
uM
XMD8-92 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-15.6
10
uM
XMD8-92 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
10.0
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
3.9
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
6.7
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
11.7
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-16.3
10
uM
XMD8-92 PC-3 AGK
ATVFLNPAACkGK
ATP
-18.4
10
uM
XMD8-92 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
40.4
10
uM
XMD8-92 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-28.7
10
uM