XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 12.5 | 10 | uM |
XMD8-92 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -12.5 | 10 | uM |
XMD8-92 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -11.9 | 10 | uM |
XMD8-92 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 11.8 | 10 | uM |
XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
XMD8-92 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -11.6 | 10 | uM |
XMD8-92 | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | -11.5 | 10 | uM |
XMD8-92 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -11.5 | 10 | uM |
XMD8-92 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -11.4 | 10 | uM |
XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
XMD8-92 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 11.1 | 10 | uM |
XMD8-92 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -11.0 | 10 | uM |
XMD8-92 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 10.9 | 10 | uM |
XMD8-92 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 10.9 | 10 | uM |
XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
XMD8-92 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 10.8 | 10 | uM |
XMD8-92 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 10.7 | 10 | uM |
XMD8-92 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 10.6 | 10 | uM |
XMD8-92 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | 10.6 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -10.5 | 10 | uM |
XMD8-92 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -10.5 | 10 | uM |
XMD8-92 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -10.4 | 10 | uM |
XMD8-92 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | -10.4 | 10 | uM |
XMD8-92 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 10.0 | 10 | uM |