XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
12.5
10
uM
XMD8-92 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-12.5
10
uM
XMD8-92 HeLa NEK9
LGDYGLAkK
Activation Loop
-11.9
10
uM
XMD8-92 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
11.8
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
11.7
10
uM
XMD8-92 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-11.6
10
uM
XMD8-92 HeLa PKR
DLkPSNIFLVDTK
Lys2
-11.5
10
uM
XMD8-92 HeLa LATS2
VDTHALYAMkTLR
Lys1
-11.5
10
uM
XMD8-92 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
-11.4
10
uM
XMD8-92 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-11.2
10
uM
XMD8-92 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-11.2
10
uM
XMD8-92 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
11.1
10
uM
XMD8-92 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-11.0
10
uM
XMD8-92 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
10.9
10
uM
XMD8-92 PC-3 MLTK
WISQDKEVAVKk
Lys1
10.9
10
uM
XMD8-92 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
-10.9
10
uM
XMD8-92 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
10.8
10
uM
XMD8-92 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
10.7
10
uM
XMD8-92 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
10.6
10
uM
XMD8-92 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
10.6
10
uM
XMD8-92 PC-3 EPHA2
EVPVAIkTLK
Lys1
-10.5
10
uM
XMD8-92 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
-10.5
10
uM
XMD8-92 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-10.4
10
uM
XMD8-92 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-10.4
10
uM
XMD8-92 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
10.0
10
uM