XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -8.6 | 10 | uM |
XMD8-92 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | 8.3 | 10 | uM |
XMD8-92 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.3 | 10 | uM |
XMD8-92 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | -8.1 | 10 | uM |
XMD8-92 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 7.9 | 10 | uM |
XMD8-92 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 7.8 | 10 | uM |
XMD8-92 | HeLa | PKD2 | DVAVkVIDK | Lys1 | 7.6 | 10 | uM |
XMD8-92 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 7.6 | 10 | uM |
XMD8-92 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | -7.6 | 10 | uM |
XMD8-92 | HeLa | IRAK3 | SHLEHQSCTINMTSSSSkHLWYMPEEYIR | Protein Kinase Domain | 7.3 | 10 | uM |
XMD8-92 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | 7.3 | 10 | uM |
XMD8-92 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 7.3 | 10 | uM |
XMD8-92 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -7.3 | 10 | uM |
XMD8-92 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 7.2 | 10 | uM |
XMD8-92 | PC-3 | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | 7.2 | 10 | uM |
XMD8-92 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -7.2 | 10 | uM |
XMD8-92 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 7.0 | 10 | uM |
XMD8-92 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 7.0 | 10 | uM |
XMD8-92 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -7.0 | 10 | uM |
XMD8-92 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -69.6 | 10 | uM |
XMD8-92 | PC-3 | MAP2K4 | MVHKPSGQIMAVkR | Lys1 | 6.9 | 10 | uM |
XMD8-92 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 6.9 | 10 | uM |
XMD8-92 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -68.4 | 10 | uM |
XMD8-92 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 6.7 | 10 | uM |