XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-8.6
10
uM
XMD8-92 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
8.3
10
uM
XMD8-92 HeLa MAP2K3
DVkPSNVLINK
Lys2
8.3
10
uM
XMD8-92 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-8.3
10
uM
XMD8-92 PC-3 CDK10
DLkVSNLLMTDK
Lys2
-8.1
10
uM
XMD8-92 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
7.9
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 HeLa PKD2
DVAVkVIDK
Lys1
7.6
10
uM
XMD8-92 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.6
10
uM
XMD8-92 PC-3 KHS1
NVHTGELAAVkIIK
Lys1
-7.6
10
uM
XMD8-92 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
7.3
10
uM
XMD8-92 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
7.3
10
uM
XMD8-92 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
10
uM
XMD8-92 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-7.3
10
uM
XMD8-92 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
7.2
10
uM
XMD8-92 PC-3 MAP2K6
DVkPSNVLINALGQVK
Lys2
7.2
10
uM
XMD8-92 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
-7.2
10
uM
XMD8-92 PC-3 LOK
DLkAGNVLMTLEGDIR
Lys2
7.0
10
uM
XMD8-92 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
7.0
10
uM
XMD8-92 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-7.0
10
uM
XMD8-92 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-69.6
10
uM
XMD8-92 PC-3 MAP2K4
MVHKPSGQIMAVkR
Lys1
6.9
10
uM
XMD8-92 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
6.9
10
uM
XMD8-92 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-68.4
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
6.7
10
uM