XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-3.7
10
uM
XMD8-92 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
-10.5
10
uM
XMD8-92 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-3.2
10
uM
XMD8-92 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-4.3
10
uM
XMD8-92 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-9.2
10
uM
XMD8-92 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-5.7
10
uM
XMD8-92 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
10.7
10
uM
XMD8-92 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-9.3
10
uM
XMD8-92 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-68.4
10
uM
XMD8-92 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
-4.6
10
uM
XMD8-92 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-25.7
10
uM
XMD8-92 HeLa SYK
ISDFGLSkALR
Activation Loop
-2.7
10
uM
XMD8-92 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-28.7
10
uM
XMD8-92 HeLa PAN3
VMDPTkILITGK
-4.5
10
uM