XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-85 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 3.5 | 10 | uM |
| XMD8-85 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | -13.6 | 10 | uM |
| XMD8-85 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -9.5 | 10 | uM |
| XMD8-85 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | -2.8 | 10 | uM |
| XMD8-85 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -23.1 | 10 | uM |
| XMD8-85 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -14.7 | 10 | uM |
| XMD8-85 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 4.4 | 10 | uM |
| XMD8-85 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | 14.9 | 10 | uM |
| XMD8-85 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -9.4 | 10 | uM |
| XMD8-85 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 14.5 | 10 | uM |
| XMD8-85 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -6.5 | 10 | uM |
| XMD8-85 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | -9.3 | 10 | uM |
| XMD8-85 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -11.2 | 10 | uM |
| XMD8-85 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -10.0 | 10 | uM |
| XMD8-85 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -22.1 | 10 | uM |
| XMD8-85 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 2.4 | 10 | uM |
| XMD8-85 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -8.2 | 10 | uM |
| XMD8-85 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -13.0 | 10 | uM |
| XMD8-85 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -7.6 | 10 | uM |
| XMD8-85 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -24.8 | 10 | uM |
| XMD8-85 | PC-3 | CDK14 | LVALkVIR | Lys1 | -7.8 | 10 | uM |
| XMD8-85 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 11.3 | 10 | uM |
| XMD8-85 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | -2.8 | 10 | uM |
| XMD8-85 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 17.1 | 10 | uM |
| XMD8-85 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -17.4 | 10 | uM |