XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
3.0
 10
uM
XMD8-85 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-13.6
 10
uM
XMD8-85 HeLa DMPK
DIkPDNILLDR
Lys2
-13.2
 10
uM
XMD8-85 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
3.6
 10
uM
XMD8-85 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
12.3
 10
uM
XMD8-85 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
31.0
 10
uM
XMD8-85 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-22.1
 10
uM
XMD8-85 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
3.8
 10
uM
XMD8-85 PC-3 EGFR
IPVAIkELR
Lys1
-6.8
 10
uM
XMD8-85 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-18.1
 10
uM
XMD8-85 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-17.1
 10
uM
XMD8-85 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
4.5
 10
uM
XMD8-85 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.3
 10
uM
XMD8-85 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
90.3
 10
uM
XMD8-85 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
12.4
 10
uM
XMD8-85 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
39.3
 10
uM
XMD8-85 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
6.2
 10
uM
XMD8-85 HeLa GCK
DTVTSELAAVkIVK
Lys1
-32.5
 10
uM
XMD8-85 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
0.0
 10
uM
XMD8-85 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-12.2
 10
uM
XMD8-85 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
5.4
 10
uM
XMD8-85 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-9.4
 10
uM
XMD8-85 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-26.4
 10
uM
XMD8-85 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
1.5
 10
uM
XMD8-85 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
9.2
 10
uM