JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
3.2
 10
uM
JWE-035 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-6.1
 10
uM
JWE-035 HeLa DMPK
DIkPDNILLDR
Lys2
-5.1
 10
uM
JWE-035 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
66.4
 10
uM
JWE-035 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
29.7
 10
uM
JWE-035 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
4.9
 10
uM
JWE-035 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.9
 10
uM
JWE-035 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.3
 10
uM
JWE-035 PC-3 EGFR
IPVAIkELR
Lys1
7.8
 10
uM
JWE-035 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
1.4
 10
uM
JWE-035 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
4.2
 10
uM
JWE-035 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
2.9
 10
uM
JWE-035 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
95.4
 10
uM
JWE-035 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
34.0
 10
uM
JWE-035 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
14.6
 10
uM
JWE-035 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
-8.1
 10
uM
JWE-035 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
41.6
 10
uM
JWE-035 HeLa GCK
DTVTSELAAVkIVK
Lys1
10.2
 10
uM
JWE-035 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.1
 10
uM
JWE-035 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-5.7
 10
uM
JWE-035 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
7.2
 10
uM
JWE-035 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-1.7
 10
uM
JWE-035 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
10.5
 10
uM
JWE-035 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
29.0
 10
uM
JWE-035 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
8.5
 10
uM