XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
85.2
 10
uM
XMD16-144 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
73.4
 10
uM
XMD16-144 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
84.2
 10
uM
XMD16-144 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
15.7
 10
uM
XMD16-144 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
16.1
 10
uM
XMD16-144 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
-16.8
 10
uM
XMD16-144 HeLa PKR
DLkPSNIFLVDTK
Lys2
-16.1
 10
uM
XMD16-144 PC-3 PKR
DLkPSNIFLVDTK
Lys2
-22.0
 10
uM
XMD16-144 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
1.8
 10
uM
XMD16-144 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
-11.8
 10
uM
XMD16-144 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-19.7
 10
uM
XMD16-144 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
12.1
 10
uM
XMD16-144 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
24.3
 10
uM
XMD16-144 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
47.5
 10
uM
XMD16-144 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
18.0
 10
uM
XMD16-144 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
54.3
 10
uM
XMD16-144 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
9.2
 10
uM
XMD16-144 HeLa SGK3
FYAVkVLQK
Lys1
3.3
 10
uM
XMD16-144 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
24.5
 10
uM
XMD16-144 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
-5.2
 10
uM
XMD16-144 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
14.6
 10
uM
XMD16-144 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
72.8
 10
uM
XMD16-144 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
 10
uM
XMD16-144 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
52.3
 10
uM
XMD16-144 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
74.3
 10
uM