XMD16-144 KiNativ -- single dose experiment
- Dataset (ID:20099)
Detail
Small Molecules Studied
Cell Lines Studied
Proteins Studied
Data Columns
Results
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Small molecules
Cells
Proteins
10091:XMD16-144
50061:HeLa
50454:PC-3
200633:ABL,ARG
200635:ACK
200636:AGK
200639:AMPKa1,AMPKa2
200640:AMPKa1,AMPKa2
200641:ARAF
200643:ATR
200647:BRAF
200648:CaMK1a
200650:CaMK2g
200653:CASK
200655:CDK10
200656:CDK11,CDK8
200658:CDK2
200661:CDK5
200663:CDK7
200664:CDK9
200666:CHK2
200667:KC1A
200668:CK1d,CK1e
200669:CSK
200671:DMPK
200672:DNAPK
200675:DNAPK
200677:eEF2K
200678:EGFR
200679:EPHA2
200681:MK03
200682:Erk5
200683:FAK
200686:FER
200687:FYN,SRC,YES
200689:GCK
200691:GCN2_domain2
200693:GSK3A
200694:GSK3B
200695:IKKA
200697:IKKE,TBK1
200698:ILK
200700:IRAK1
200701:IRAK4
200702:IRE1
200704:JAK1
200705:JAK1_domain2
200706:JAK1_domain2
200707:JNK1,JNK2,JNK3
200710:KHS1
200711:LATS1
200712:LKB1
200714:LOK
200716:LOK
200719:MAP2K1,MAP2K2
200722:MAP2K3
200723:MAP2K4
200724:MAP2K4
200726:MAP2K6
200728:MAP2K6
200730:MAP3K1
200731:M3K2
200732:M3K2,MAP3K3
200734:MAP3K4
200735:MAP3K5,MAP3K6,MAP3K7
200739:MARK2,MARK3
200742:MAST2,MAST4
200743:MAST3
200746:MLK3
200748:MPSK1
200749:MSK1,MSK2_domain1
200750:MSK1_domain1
200751:MST1
200753:MST1,MST2
200755:MST2
200756:MST3
200759:MST4,YSK1
200764:NDR2
200767:NEK1
200768:NEK6,NEK7
200771:NEK8
200774:NEK9
200775:NEK9
200777:p38d,p38g
200779:KS6B1
200780:p70S6K,p70S6Kb
200782:KS6B2
200783:CDK16
200784:PCTAIRE2
200787:CDK14
200788:PHKg2
200789:PI4KA,PI4KAP2
200790:PI4KB
200793:PIK3C3
200795:PIK3CB
200799:PI42C
200801:PITSLRE
200802:PKCa,PKCb
200805:PKD1,PKD2
200809:PKR
200812:PRPK
200814:ROCK1,ROCK2
200816:RSK1,RSK2_domain1
200820:RSK2_domain1
200821:RSK2_domain2
200822:RSK2_domain2
200825:RSKL1_domain1
200826:SGK3
200829:SLK
200830:SMG1
200832:SRC
200833:STLK5
200834:TAO1,TAOK3
200835:TAOK2
200836:TBK1
200837:TLK1
200838:TLK2
200841:WEE1
200842:Wnk1,Wnk2,Wnk3
200843:Wnk1,Wnk2,Wnk4
200844:WNK4
200845:MLTK
200847:ZC1/HGK,ZC2/TNIK,ZC3/MINK
200877:BARK1
200880:BTK
200882:CAMK1D
200890:CDK5
200895:CHK1
200896:CHK2
200907:DGKA
200911:EPHB4
200916:FES
200928:HPK1
200933:IKKE
200937:KSR1,KSR2
200938:LATS2
200940:LYN
200943:M3K2
200944:MAP3K5
200945:MAPKAPK3
200947:MARK2
200949:MARK3,MARK4
200950:MASTL
200951:MET
200952:MRCKb
200965:p38a
200967:MK14
200969:PAN3
200973:PEK
200978:PIK3CG
200989:PKN1
200992:PLK1
201002:ROCK1
201003:RON
201013:SRPK1
201014:SRPK1/2
201026:ULK3
201035:EGFR
201041:KPCI
201043:PRP4
201046:ANPb
201047:CaMK2a,CaMK2b,CaMK2d,CaMK2g
201048:CDK5
201049:CK2a2
201050:EGFR
201051:EphA1
201052:EPHA2
201053:EphA7
201054:EPHB2
201055:GCN2
201056:JAK2 domain2
201057:JAK3 domain2
201058:M4K3
201059:MET
201060:MRCKb
201061:MK11
201062:PDK1
201063:PI42C
201064:PKD2
201065:RIPK3
201066:RSK1 domain1
201067:RSK1,RSK4 domain1
201068:SLK
201069:SYK
201070:TLK1
201071:ULK1
201072:AurB
201073:CLK2
201074:IRAK3
201075:MYO3A,MYO3B
201076:SNRK
201077:TEC
201078:ILK
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Small Molecule
Cell Line
Protein
Sequence
Labeling Site
% Inhibition
Assay compound conc
Conc unit
XMD16-144
HeLa
RIPK3
DLkPSNVLLDPELHVK
Lys2
-3.7
10
uM
XMD16-144
HeLa
RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-4.7
10
uM
XMD16-144
HeLa
RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
10.2
10
uM
XMD16-144
PC-3
SLK
ETSVLAAAkVIDTK
Lys1
33.2
10
uM
XMD16-144
HeLa
SYK
ISDFGLSkALR
Activation Loop
14.5
10
uM
XMD16-144
HeLa
TLK1
YAAVkIHQLNK
Lys1
14.3
10
uM
XMD16-144
PC-3
TLK1
YAAVkIHQLNK
Lys1
-10.1
10
uM
XMD16-144
HeLa
ULK1
DLkPQNILLSNPAGR
Lys2
-15.7
10
uM
XMD16-144
HeLa
AurB
SHFIVALkVLFK
Lys1
97.3
10
uM
XMD16-144
PC-3
CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
10.0
10
uM
XMD16-144
HeLa
IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
19.2
10
uM
XMD16-144
HeLa
MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-7.1
10
uM
XMD16-144
PC-3
SNRK
DLkPENVVFFEK
Lys2
-8.0
10
uM
XMD16-144
HeLa
TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
27.3
10
uM
XMD16-144
HeLa
ILK
WQGIVVkVLK
Lys1
1.0
10
uM
XMD16-144
PC-3
ILK
WQGIVVkVLK
Lys1
3.0
10
uM
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