XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD16-144 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 14.9 | 10 | uM |
| XMD16-144 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -2.5 | 10 | uM |
| XMD16-144 | HeLa | KPCI | IYAMkVVK | Lys1 | -20.5 | 10 | uM |
| XMD16-144 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | 4.1 | 10 | uM |
| XMD16-144 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -30.6 | 10 | uM |
| XMD16-144 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 42.2 | 10 | uM |
| XMD16-144 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -2.8 | 10 | uM |
| XMD16-144 | PC-3 | CK2a2 | DVkPHNVMIDHQQK | Lys2 | 20.2 | 10 | uM |
| XMD16-144 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -7.5 | 10 | uM |
| XMD16-144 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 41.9 | 10 | uM |
| XMD16-144 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | 27.8 | 10 | uM |
| XMD16-144 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 11.1 | 10 | uM |
| XMD16-144 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 43.9 | 10 | uM |
| XMD16-144 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -4.9 | 10 | uM |
| XMD16-144 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 3.3 | 10 | uM |
| XMD16-144 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 4.5 | 10 | uM |
| XMD16-144 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -48.5 | 10 | uM |
| XMD16-144 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 44.1 | 10 | uM |
| XMD16-144 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 57.2 | 10 | uM |
| XMD16-144 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 8.9 | 10 | uM |
| XMD16-144 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 4.7 | 10 | uM |
| XMD16-144 | PC-3 | PDK1 | EYAIkILEK | Lys1 | 7.7 | 10 | uM |
| XMD16-144 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 54.0 | 10 | uM |
| XMD16-144 | HeLa | PKD2 | DVAVkVIDK | Lys1 | -8.8 | 10 | uM |
| XMD16-144 | PC-3 | PKD2 | DVAVkVIDK | Lys1 | 31.0 | 10 | uM |