XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD16-144 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -14.4 | 10 | uM |
XMD16-144 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -10.3 | 10 | uM |
XMD16-144 | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | 14.3 | 10 | uM |
XMD16-144 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 61.5 | 10 | uM |
XMD16-144 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | 2.1 | 10 | uM |
XMD16-144 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 11.8 | 10 | uM |
XMD16-144 | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | 75.9 | 10 | uM |
XMD16-144 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | 81.2 | 10 | uM |
XMD16-144 | HeLa | MASTL | LYAVkVVK | Lys1 | 26.9 | 10 | uM |
XMD16-144 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 0.2 | 10 | uM |
XMD16-144 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | -22.5 | 10 | uM |
XMD16-144 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -7.7 | 10 | uM |
XMD16-144 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | 24.3 | 10 | uM |
XMD16-144 | HeLa | MK14 | QELNkTIWEVPER | Other | 4.0 | 10 | uM |
XMD16-144 | PC-3 | MK14 | QELNkTIWEVPER | Other | -30.0 | 10 | uM |
XMD16-144 | HeLa | PAN3 | VMDPTkILITGK | -12.8 | 10 | uM | |
XMD16-144 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -33.3 | 10 | uM |
XMD16-144 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | -9.1 | 10 | uM |
XMD16-144 | HeLa | PIK3CG | KkPLWLEFK | ATP | 14.3 | 10 | uM |
XMD16-144 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | -5.0 | 10 | uM |
XMD16-144 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | -0.9 | 10 | uM |
XMD16-144 | PC-3 | ROCK1 | kLQLELNQER | Other | 3.5 | 10 | uM |
XMD16-144 | PC-3 | RON | IQCAIkSLSR | Lys1 | -1.2 | 10 | uM |
XMD16-144 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | -6.0 | 10 | uM |
XMD16-144 | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | 1.8 | 10 | uM |