XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -15.8 | 10 | uM |
XMD11-85h | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -1.8 | 10 | uM |
XMD11-85h | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | -1.7 | 10 | uM |
XMD11-85h | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | -4.5 | 10 | uM |
XMD11-85h | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -2.9 | 10 | uM |
XMD11-85h | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 3.0 | 10 | uM |
XMD11-85h | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 16.4 | 10 | uM |
XMD11-85h | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | -3.4 | 10 | uM |
XMD11-85h | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -3.4 | 10 | uM |
XMD11-85h | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -5.1 | 10 | uM |
XMD11-85h | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | -28.4 | 10 | uM |
XMD11-85h | HeLa | MLTK | WISQDKEVAVKk | Lys1 | -37.6 | 10 | uM |
XMD11-85h | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 8.5 | 10 | uM |
XMD11-85h | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -14.1 | 10 | uM |
XMD11-85h | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -15.3 | 10 | uM |
XMD11-85h | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -33.3 | 10 | uM |
XMD11-85h | HeLa | BTK | GQYDVAIkMIK | Lys1 | -35.0 | 10 | uM |
XMD11-85h | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -8.9 | 10 | uM |
XMD11-85h | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 0.6 | 10 | uM |
XMD11-85h | HeLa | CHK1 | DIkPENLLLDER | Lys2 | -11.0 | 10 | uM |
XMD11-85h | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -20.1 | 10 | uM |
XMD11-85h | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 3.8 | 10 | uM |
XMD11-85h | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | 60.9 | 10 | uM |
XMD11-85h | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 0.4 | 10 | uM |
XMD11-85h | HeLa | FES | LRADNTLVAVkSCR | Lys1 | -8.4 | 10 | uM |