XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-15.8
10
uM
XMD11-85h PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-1.8
10
uM
XMD11-85h PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
-1.7
10
uM
XMD11-85h HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
-4.5
10
uM
XMD11-85h HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-2.9
10
uM
XMD11-85h PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
3.0
10
uM
XMD11-85h PC-3 TLK2
YVAVkIHQLNK
Lys1
16.4
10
uM
XMD11-85h HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-3.4
10
uM
XMD11-85h HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-3.4
10
uM
XMD11-85h PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-5.1
10
uM
XMD11-85h PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-28.4
10
uM
XMD11-85h HeLa MLTK
WISQDKEVAVKk
Lys1
-37.6
10
uM
XMD11-85h PC-3 MLTK
WISQDKEVAVKk
Lys1
8.5
10
uM
XMD11-85h HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-14.1
10
uM
XMD11-85h PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-15.3
10
uM
XMD11-85h HeLa BARK1
DLkPANILLDEHGHVR
Lys2
-33.3
10
uM
XMD11-85h HeLa BTK
GQYDVAIkMIK
Lys1
-35.0
10
uM
XMD11-85h HeLa CAMK1D
LFAVkCIPK
Lys1
-8.9
10
uM
XMD11-85h PC-3 CDK5
DLkPQNLLINR
Lys2
0.6
10
uM
XMD11-85h HeLa CHK1
DIkPENLLLDER
Lys2
-11.0
10
uM
XMD11-85h HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
-20.1
10
uM
XMD11-85h PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
3.8
10
uM
XMD11-85h HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
60.9
10
uM
XMD11-85h PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
0.4
10
uM
XMD11-85h HeLa FES
LRADNTLVAVkSCR
Lys1
-8.4
10
uM