XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h PC-3 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
1.6
10
uM
XMD11-85h HeLa MST3
DIkAANVLLSEHGEVK
Lys2
-12.1
10
uM
XMD11-85h PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
-15.3
10
uM
XMD11-85h PC-3 NDR2
DTGHIYAMkILR
Lys1
2.6
10
uM
XMD11-85h HeLa NEK1
DIkSQNIFLTK
Lys2
-19.6
10
uM
XMD11-85h HeLa NEK6,NEK7
DIkPANVFITATGVVK
Lys2
1.4
10
uM
XMD11-85h PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
2.6
10
uM
XMD11-85h PC-3 NEK8
DLkTQNILLDK
Lys2
19.9
10
uM
XMD11-85h HeLa NEK9
DIkTLNIFLTK
Lys2
2.9
10
uM
XMD11-85h PC-3 NEK9
DIkTLNIFLTK
Lys2
4.7
10
uM
XMD11-85h HeLa NEK9
LGDYGLAkK
Activation Loop
-20.3
10
uM
XMD11-85h PC-3 NEK9
LGDYGLAkK
Activation Loop
7.8
10
uM
XMD11-85h HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-37.3
10
uM
XMD11-85h PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-18.2
10
uM
XMD11-85h HeLa KS6B1
DLkPENIMLNHQGHVK
Lys2
-30.4
10
uM
XMD11-85h PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
26.1
10
uM
XMD11-85h PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-6.0
10
uM
XMD11-85h HeLa KS6B2
DLkPENIMLSSQGHIK
Lys2
-26.0
10
uM
XMD11-85h PC-3 CDK16
LTDNLVALkEIR
Lys1
-12.2
10
uM
XMD11-85h HeLa PCTAIRE2
DLkPQNLLINEK
Lys2
-22.0
10
uM
XMD11-85h PC-3 CDK14
LVALkVIR
Lys1
-22.4
10
uM
XMD11-85h PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
20.8
10
uM
XMD11-85h HeLa PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
-22.7
10
uM
XMD11-85h PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
8.6
10
uM
XMD11-85h HeLa PI4KB
VPHTQAVVLNSkDK
ATP
-20.8
10
uM