XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 1.6 | 10 | uM |
XMD11-85h | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | -12.1 | 10 | uM |
XMD11-85h | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -15.3 | 10 | uM |
XMD11-85h | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 2.6 | 10 | uM |
XMD11-85h | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -19.6 | 10 | uM |
XMD11-85h | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 1.4 | 10 | uM |
XMD11-85h | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 2.6 | 10 | uM |
XMD11-85h | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | 19.9 | 10 | uM |
XMD11-85h | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | 2.9 | 10 | uM |
XMD11-85h | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 4.7 | 10 | uM |
XMD11-85h | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -20.3 | 10 | uM |
XMD11-85h | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 7.8 | 10 | uM |
XMD11-85h | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -37.3 | 10 | uM |
XMD11-85h | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -18.2 | 10 | uM |
XMD11-85h | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -30.4 | 10 | uM |
XMD11-85h | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 26.1 | 10 | uM |
XMD11-85h | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -6.0 | 10 | uM |
XMD11-85h | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -26.0 | 10 | uM |
XMD11-85h | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -12.2 | 10 | uM |
XMD11-85h | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -22.0 | 10 | uM |
XMD11-85h | PC-3 | CDK14 | LVALkVIR | Lys1 | -22.4 | 10 | uM |
XMD11-85h | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 20.8 | 10 | uM |
XMD11-85h | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | -22.7 | 10 | uM |
XMD11-85h | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 8.6 | 10 | uM |
XMD11-85h | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -20.8 | 10 | uM |