XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -2.4 | 10 | uM |
XMD11-50 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -1.9 | 10 | uM |
XMD11-50 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -11.2 | 10 | uM |
XMD11-50 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 13.2 | 10 | uM |
XMD11-50 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 6.4 | 10 | uM |
XMD11-50 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 6.5 | 10 | uM |
XMD11-50 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -18.4 | 10 | uM |
XMD11-50 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.3 | 10 | uM |
XMD11-50 | PC-3 | EGFR | IPVAIkELR | Lys1 | 1.4 | 10 | uM |
XMD11-50 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -4.8 | 10 | uM |
XMD11-50 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -1.1 | 10 | uM |
XMD11-50 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 10.8 | 10 | uM |
XMD11-50 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.8 | 10 | uM |
XMD11-50 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 60.0 | 10 | uM |
XMD11-50 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 35.0 | 10 | uM |
XMD11-50 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 25.4 | 10 | uM |
XMD11-50 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 7.2 | 10 | uM |
XMD11-50 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 11.9 | 10 | uM |
XMD11-50 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 3.8 | 10 | uM |
XMD11-50 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | 1.3 | 10 | uM |
XMD11-50 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 10.1 | 10 | uM |
XMD11-50 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.5 | 10 | uM |
XMD11-50 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -0.2 | 10 | uM |
XMD11-50 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | -14.2 | 10 | uM |
XMD11-50 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 3.8 | 10 | uM |