XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-2.4
10
uM
XMD11-50 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-1.9
10
uM
XMD11-50 HeLa DMPK
DIkPDNILLDR
Lys2
-11.2
10
uM
XMD11-50 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
13.2
10
uM
XMD11-50 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
6.4
10
uM
XMD11-50 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
6.5
10
uM
XMD11-50 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-18.4
10
uM
XMD11-50 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-5.3
10
uM
XMD11-50 PC-3 EGFR
IPVAIkELR
Lys1
1.4
10
uM
XMD11-50 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-4.8
10
uM
XMD11-50 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-1.1
10
uM
XMD11-50 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
10.8
10
uM
XMD11-50 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.8
10
uM
XMD11-50 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
60.0
10
uM
XMD11-50 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
35.0
10
uM
XMD11-50 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
25.4
10
uM
XMD11-50 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
7.2
10
uM
XMD11-50 HeLa GCK
DTVTSELAAVkIVK
Lys1
11.9
10
uM
XMD11-50 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
3.8
10
uM
XMD11-50 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
1.3
10
uM
XMD11-50 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
10.1
10
uM
XMD11-50 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-7.5
10
uM
XMD11-50 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-0.2
10
uM
XMD11-50 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
-14.2
10
uM
XMD11-50 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
3.8
10
uM