PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)
Proteins Studied
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LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200704 | JAK1 | 200704 | P23458 | Tyrosine-protein kinase JAK1 | KiNativ | ||||
200705 | JAK1_domain2 | 200705 | P23458 | Tyrosine-protein kinase JAK1 | KiNativ | domain2 | |||
200658 | CDK2 | 200658 | P24941 | Cyclin-dependent kinase 2; p33 protein kinase | KiNativ | ||||
200657 | CDK2 | 200657 | P24941 | Cyclin-dependent kinase 2; p33 protein kinase | KiNativ | ||||
200681 | MK03 | 200681 | P27361 | Mitogen-activated protein kinase 3 | KiNativ | ||||
200680 | MK03 | 200680 | P27361 | Mitogen-activated protein kinase 3 | KiNativ | ||||
200740 | MARK3 | 200740 | P27448 | MAP/microtubule affinity-regulating kinase 3 | KiNativ | ||||
200739 | MARK2,MARK3 | 200739 | P27448 | MAP/microtubule affinity-regulating kinase 3 | KiNativ | ||||
200679 | EPHA2 | 200679 | P29317 | Ephrin type-A receptor 2 | KiNativ | ||||
200841 | WEE1 | 200841 | P30291 | Wee1-like protein kinase; DKFZp686I18166; FLJ16446; WEE1; WEE1A; WEE1hu | KiNativ | ||||
200646 | AXL | 200646 | P30530 | Tyrosine-protein kinase receptor UFO precursor | KiNativ | ||||
200637 | AKT1 | 200637 | P31749 | V-akt murine thymoma viral oncogene homolog 1; AKT; AKT1; Akt1/PKBa; MGC99656; PKB; PKBa; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA | KiNativ | ||||
200638 | AKT2,AKT3 | 200638 | P31751 | RAC-beta serine/threonine-protein kinase | KiNativ | ||||
200669 | CSK | 200669 | P41240 | Tyrosine-protein kinase CSK | KiNativ | ||||
200670 | CSK | 200670 | P41240 | Tyrosine-protein kinase CSK | KiNativ | ||||
200794 | PIK3CA | 200794 | P42336 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha | KiNativ | ||||
200795 | PIK3CB | 200795 | P42338 | Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit beta; DKFZp779K1237; MGC133043; P110BETA; PI3K; PI3KBETA; PIK3C1; PIK3CB; PI3K-beta | KiNativ | ||||
200789 | PI4KA,PI4KAP2 | 200789 | P42356 | Phosphatidylinositol 4-kinase alpha | KiNativ | ||||
200707 | JNK1,JNK2,JNK3 | 200707 | P45983 | Mitogen-activated protein kinase 8 | KiNativ | ||||
200723 | MAP2K4 | 200723 | P45985 | Dual specificity mitogen-activated protein kinase kinase 4 | KiNativ | ||||
200724 | MAP2K4 | 200724 | P45985 | Dual specificity mitogen-activated protein kinase kinase 4 | KiNativ | ||||
200722 | MAP2K3 | 200722 | P46734 | Dual specificity mitogen-activated protein kinase kinase 3 | KiNativ | ||||
200797 | PIP4K2A | 200797 | P48426 | Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha; 1-phosphatidylinositol 5-phosphate 4-kinase 2-alpha; Diphosphoinositide kinase 2-alpha; PIP5KIII | KiNativ | ||||
200667 | KC1A | 200667 | P48729 | Casein kinase I isoform alpha | KiNativ | ||||
200668 | CK1d,CK1e | 200668 | P48730 | Casein kinase I isoform delta | KiNativ |