PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200704 JAK1 200704 P23458
Tyrosine-protein kinase JAK1
KiNativ
200705 JAK1_domain2 200705 P23458
Tyrosine-protein kinase JAK1
KiNativ domain2
200658 CDK2 200658 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200657 CDK2 200657 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200681 MK03 200681 P27361
Mitogen-activated protein kinase 3
KiNativ
200680 MK03 200680 P27361
Mitogen-activated protein kinase 3
KiNativ
200740 MARK3 200740 P27448
MAP/microtubule affinity-regulating kinase 3
KiNativ
200739 MARK2,MARK3 200739 P27448
MAP/microtubule affinity-regulating kinase 3
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
200841 WEE1 200841 P30291
Wee1-like protein kinase; DKFZp686I18166; FLJ16446; WEE1; WEE1A; WEE1hu
KiNativ
200646 AXL 200646 P30530
Tyrosine-protein kinase receptor UFO precursor
KiNativ
200637 AKT1 200637 P31749
V-akt murine thymoma viral oncogene homolog 1; AKT; AKT1; Akt1/PKBa; MGC99656; PKB; PKBa; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA
KiNativ
200638 AKT2,AKT3 200638 P31751
RAC-beta serine/threonine-protein kinase
KiNativ
200669 CSK 200669 P41240
Tyrosine-protein kinase CSK
KiNativ
200670 CSK 200670 P41240
Tyrosine-protein kinase CSK
KiNativ
200794 PIK3CA 200794 P42336
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit alpha; MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA; PI3K-alpha
KiNativ
200795 PIK3CB 200795 P42338
Phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit beta; DKFZp779K1237; MGC133043; P110BETA; PI3K; PI3KBETA; PIK3C1; PIK3CB; PI3K-beta
KiNativ
200789 PI4KA,PI4KAP2 200789 P42356
Phosphatidylinositol 4-kinase alpha
KiNativ
200707 JNK1,JNK2,JNK3 200707 P45983
Mitogen-activated protein kinase 8
KiNativ
200723 MAP2K4 200723 P45985
Dual specificity mitogen-activated protein kinase kinase 4
KiNativ
200724 MAP2K4 200724 P45985
Dual specificity mitogen-activated protein kinase kinase 4
KiNativ
200722 MAP2K3 200722 P46734
Dual specificity mitogen-activated protein kinase kinase 3
KiNativ
200797 PIP4K2A 200797 P48426
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha; 1-phosphatidylinositol 5-phosphate 4-kinase 2-alpha; Diphosphoinositide kinase 2-alpha; PIP5KIII
KiNativ
200667 KC1A 200667 P48729
Casein kinase I isoform alpha
KiNativ
200668 CK1d,CK1e 200668 P48730
Casein kinase I isoform delta
KiNativ