PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200711 LATS1 200711 O95835
Serine/threonine-protein kinase LATS1
KiNativ
200666 CHK2 200666 O96017
Serine/threonine-protein kinase Chk2; CHK2 checkpoint homolog
KiNativ
200634 ABL,ARG 200634 P00519
Proto-oncogene tyrosine-protein kinase ABL1
KiNativ
200633 ABL,ARG 200633 P00519
Proto-oncogene tyrosine-protein kinase ABL1
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
200813 RAF1 200813 P04049
RAF proto-oncogene serine/threonine-protein kinase; CRAF; c-Raf; NS5; RAF1; Raf-1
KiNativ
200687 FYN,SRC,YES 200687 P06241
Proto-oncogene tyrosine-protein kinase Fyn
KiNativ
200654 CDC2 200654 P06493
Cell division control protein 2 homolog
KiNativ
200641 ARAF 200641 P10398
A-Raf proto-oncogene serine/threonine-protein kinase
KiNativ
200659 CDK4 200659 P11802
Cyclin-dependent kinase 4; cell division protein kinase 4
KiNativ
200831 SRC 200831 P12931
Proto-oncogene tyrosine-protein kinase Src; V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian); ASV; c-SRC; p60-Src; SRC; SRC1
KiNativ
200832 SRC 200832 P12931
Proto-oncogene tyrosine-protein kinase Src; V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian); ASV; c-SRC; p60-Src; SRC; SRC1
KiNativ
200647 BRAF 200647 P15056
Serine/threonine-protein kinase B-raf; v-raf murine sarcoma viral oncogene homolog B1; BRAF1; RAFB1
KiNativ
200788 PHKg2 200788 P15735
Phosphorylase b kinase gamma catalytic chain, testis/liver isoform
KiNativ
200685 FER 200685 P16591
Proto-oncogene tyrosine-protein kinase FER
KiNativ
200684 FER 200684 P16591
Proto-oncogene tyrosine-protein kinase FER
KiNativ
200686 FER 200686 P16591
Proto-oncogene tyrosine-protein kinase FER
KiNativ
200802 PKCa,PKCb 200802 P17252
Protein kinase C alpha type
KiNativ
200809 PKR 200809 P19525
Interferon-induced, double-stranded RNA-activated protein kinase
KiNativ
200801 PITSLRE 200801 P21127
PITSLRE serine/threonine-protein kinase CDC2L1
KiNativ
200811 PRKACB 200811 P22694
CAMP-dependent protein kinase catalytic subunit beta
KiNativ
200778 KS6B1 200778 P23443
Ribosomal protein S6 kinase 1 (EC 2.7.1.37) (S6K) (S6K1) (70 kDa ribosomal protein S6 kinase 1) (p70 S6 kinase alpha) (p70(S6K)-alpha)
KiNativ
200780 p70S6K,p70S6Kb 200780 P23443
Ribosomal protein S6 kinase 1 (EC 2.7.1.37) (S6K) (S6K1) (70 kDa ribosomal protein S6 kinase 1) (p70 S6 kinase alpha) (p70(S6K)-alpha)
KiNativ
200779 KS6B1 200779 P23443
Ribosomal protein S6 kinase 1 (EC 2.7.1.37) (S6K) (S6K1) (70 kDa ribosomal protein S6 kinase 1) (p70 S6 kinase alpha) (p70(S6K)-alpha)
KiNativ
200704 JAK1 200704 P23458
Tyrosine-protein kinase JAK1
KiNativ