PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200658 CDK2 200658 P24941
Cyclin-dependent kinase 2; p33 protein kinase
KiNativ
200659 CDK4 200659 P11802
Cyclin-dependent kinase 4; cell division protein kinase 4
KiNativ
200660 CDK5 200660 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
200661 CDK5 200661 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KiNativ
200662 CDK6 200662 Q00534
Cyclin-dependent kinase 6; cell division protein kinase 6
KiNativ
200633 ABL,ARG 200633 P00519
Proto-oncogene tyrosine-protein kinase ABL1
KiNativ
200644 AurA 200644 O14965
Serine/threonine-protein kinase 6
KiNativ
200654 CDC2 200654 P06493
Cell division control protein 2 homolog
KiNativ
200653 CASK 200653 O14936
Peripheral plasma membrane protein CASK
KiNativ
200638 AKT2,AKT3 200638 P31751
RAC-beta serine/threonine-protein kinase
KiNativ
200652 CaMKK2 200652 Q96RR4
Calcium/calmodulin-dependent protein kinase kinase 2
KiNativ
200672 DNAPK 200672 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200671 DMPK 200671 Q09013
Myotonin-protein kinase; Dystrophia myotonica-protein kinase; DM; DM1; DM1PK; DMK; MDPK; MT-PK
KiNativ
200651 CaMK2g 200651 Q13555
Calcium/calmodulin-dependent protein kinase type II gamma chain
KiNativ
200637 AKT1 200637 P31749
V-akt murine thymoma viral oncogene homolog 1; AKT; AKT1; Akt1/PKBa; MGC99656; PKB; PKBa; PKB-ALPHA; PRKBA; RAC; RAC-ALPHA
KiNativ
200673 DNAPK 200673 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200772 NEK9 200772 Q8TD19
Serine/threonine-protein kinase Nek9
KiNativ
200674 DNAPK 200674 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200675 DNAPK 200675 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200676 eEF2K 200676 O00418
Elongation factor 2 kinase
KiNativ
200677 eEF2K 200677 O00418
Elongation factor 2 kinase
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
200771 NEK8 200771 Q86SG6
Serine/threonine-protein kinase Nek8
KiNativ
200670 CSK 200670 P41240
Tyrosine-protein kinase CSK
KiNativ