PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200662 CDK6 200662 Q00534
Cyclin-dependent kinase 6; cell division protein kinase 6
KiNativ
200663 CDK7 200663 P50613
Cyclin-dependent kinase 7; cell division protein kinase 7; CAK1; CDK7; CDKN7; MO15; p39MO15; STK1
KiNativ
200664 CDK9 200664 P50750
Cyclin-dependent kinase 9; cell division protein kinase 9; C-2k; CDC2L4; CDK9; CTK1; PITALRE; TAK
KiNativ
200675 DNAPK 200675 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200674 DNAPK 200674 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200673 DNAPK 200673 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200672 DNAPK 200672 P78527
DNA-dependent protein kinase catalytic subunit
KiNativ
200718 MAP2K1 200718 Q02750
Dual specificity mitogen-activated protein kinase kinase 1
KiNativ
200719 MAP2K1,MAP2K2 200719 Q02750
Dual specificity mitogen-activated protein kinase kinase 1
KiNativ
200720 MAP2K1,MAP2K2 200720 Q02750
Dual specificity mitogen-activated protein kinase kinase 1
KiNativ
200721 MAP2K1,MAP2K2 200721 Q02750
Dual specificity mitogen-activated protein kinase kinase 1
KiNativ
200722 MAP2K3 200722 P46734
Dual specificity mitogen-activated protein kinase kinase 3
KiNativ
200724 MAP2K4 200724 P45985
Dual specificity mitogen-activated protein kinase kinase 4
KiNativ
200723 MAP2K4 200723 P45985
Dual specificity mitogen-activated protein kinase kinase 4
KiNativ
200725 MAP2K5 200725 Q13163
Dual specificity mitogen-activated protein kinase kinase 5
KiNativ
200726 MAP2K6 200726 P52564
Dual specificity mitogen-activated protein kinase kinase 6
KiNativ
200728 MAP2K6 200728 P52564
Dual specificity mitogen-activated protein kinase kinase 6
KiNativ
200727 MAP2K6 200727 P52564
Dual specificity mitogen-activated protein kinase kinase 6
KiNativ
200729 MP2K7 200729 O14733
Dual specificity mitogen-activated protein kinase kinase 7
KiNativ
200677 eEF2K 200677 O00418
Elongation factor 2 kinase
KiNativ
200676 eEF2K 200676 O00418
Elongation factor 2 kinase
KiNativ
200679 EPHA2 200679 P29317
Ephrin type-A receptor 2
KiNativ
200678 EGFR 200678 P00533
Epidermal growth factor receptor precursor
KiNativ
200692 GCN2_domain2 200692 Q9P2K8
Eukaryotic translation initiation factor 2-alpha kinase 4
KiNativ domain2
200691 GCN2_domain2 200691 Q9P2K8
Eukaryotic translation initiation factor 2-alpha kinase 4
KiNativ domain2