PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200808 PKN2 200808 Q16513
Protein kinase N2
KiNativ
200809 PKR 200809 P19525
Interferon-induced, double-stranded RNA-activated protein kinase
KiNativ
200810 PLK1 200810 P53350
Serine/threonine-protein kinase PLK1; polo-like kinase 1 (Drosophila); PLK; PLK1; STPK13
KiNativ
200811 PRKACB 200811 P22694
CAMP-dependent protein kinase catalytic subunit beta
KiNativ
200812 PRPK 200812 Q96S44
TP53-regulating kinase
KiNativ
200813 RAF1 200813 P04049
RAF proto-oncogene serine/threonine-protein kinase; CRAF; c-Raf; NS5; RAF1; Raf-1
KiNativ
200814 ROCK1,ROCK2 200814 O75116
Rho-associated protein kinase 2
KiNativ
200815 RSK1,RSK2,RSK3_domain1 200815 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KiNativ domain1
200816 RSK1,RSK2_domain1 200816 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KiNativ domain1
200817 RSK1_domain1 200817 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KiNativ domain1
200818 RSK1_domain1 200818 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KiNativ domain1
200819 RSK1_domain2 200819 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KiNativ domain2
200820 RSK2_domain1 200820 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KiNativ domain1
200821 RSK2_domain2 200821 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KiNativ domain2
200822 RSK2_domain2 200822 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KiNativ domain2
200823 RSK2_domain2 200823 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KiNativ domain2
200824 RSK3_domain1 200824 Q15349
Ribosomal protein S6 kinase alpha-2; S6K-alpha-2; KS6A2; p90-RSK 2; MAPKAPK-1c; pp90RSK3
KiNativ domain1
200825 RSKL1_domain1 200825 Q96S38
Ribosomal protein S6 kinase delta-1
KiNativ domain1
200826 SGK3 200826 Q96BR1
Serine/threonine-protein kinase Sgk3; Serum/glucocorticoid-regulated kinase 3; CISK; DKFZp781N0293; SGKL
KiNativ
200827 SLK 200827 Q9H2G2
STE20-like serine/threonine-protein kinase; CTCL tumor antigen se20-9; bA16H23.1; KIAA0204; LOSK; MGC133067; se20-9; SLK; STK2
KiNativ
200828 SLK 200828 Q9H2G2
STE20-like serine/threonine-protein kinase; CTCL tumor antigen se20-9; bA16H23.1; KIAA0204; LOSK; MGC133067; se20-9; SLK; STK2
KiNativ
200829 SLK 200829 Q9H2G2
STE20-like serine/threonine-protein kinase; CTCL tumor antigen se20-9; bA16H23.1; KIAA0204; LOSK; MGC133067; se20-9; SLK; STK2
KiNativ
200830 SMG1 200830 Q96Q15
Serine/threonine-protein kinase SMG1
KiNativ
200831 SRC 200831 P12931
Proto-oncogene tyrosine-protein kinase Src; V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian); ASV; c-SRC; p60-Src; SRC; SRC1
KiNativ
200832 SRC 200832 P12931
Proto-oncogene tyrosine-protein kinase Src; V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian); ASV; c-SRC; p60-Src; SRC; SRC1
KiNativ