GW-5074 KINOMEscan - Dataset (ID:20022)

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Small Molecule Protein % Control Assay compound conc Conc unit
GW-5074 AAK1 5.2 10
uM
GW-5074 ABL1(E255K)-phosphorylated 54.0 10
uM
GW-5074 ABL1(F317I)-nonphosphorylated 70.0 10
uM
GW-5074 ABL1(F317I)-phosphorylated 85.0 10
uM
GW-5074 ABL1(F317L)-nonphosphorylated 69.0 10
uM
GW-5074 ABL1(F317L)-phosphorylated 52.0 10
uM
GW-5074 ABL1(H396P)-nonphosphorylated 24.0 10
uM
GW-5074 ABL1(H396P)-phosphorylated 77.0 10
uM
GW-5074 ABL1(M351T)-phosphorylated 77.0 10
uM
GW-5074 ABL1(Q252H)-nonphosphorylated 38.0 10
uM
GW-5074 ABL1(Q252H)-phosphorylated 69.0 10
uM
GW-5074 ABL1(T315I)-nonphosphorylated 88.0 10
uM
GW-5074 ABL1(T315I)-phosphorylated 100.0 10
uM
GW-5074 ABL1(Y253F)-phosphorylated 81.0 10
uM
GW-5074 ABL1-nonphosphorylated 57.0 10
uM
GW-5074 ABL1-phosphorylated 68.0 10
uM
GW-5074 ABL2 66.0 10
uM
GW-5074 ACVR1 31.0 10
uM
GW-5074 ACVR1B 33.0 10
uM
GW-5074 ACVR2A 100.0 10
uM
GW-5074 ACVR2B 83.0 10
uM
GW-5074 ACVRL1 100.0 10
uM
GW-5074 ADCK3 100.0 10
uM
GW-5074 ADCK4 65.0 10
uM
GW-5074 AKT1 100.0 10
uM
  • Page 1 of 18
  • 1 to 25 of 442 records