Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
KIN001-269
558
1
AXL
Vandetanib
558
2
AXL
Vandetanib
558
2
AXL
RAF 265
558
10
AXL
RAF 265
558
10
AXL
JNK-IN-5A
558
10
AXL
BMS-536924
558
2
AXL
KIN001-021
558
10
AXL
PKC412
558
2
AXL
PKC412
558
2
AXL
Tofacitinib
558
10
AXL
Tofacitinib
558
10
AXL
Tofacitinib
558
10
AXL
KU63794
558
10
AXL
Lestaurtinib
558
1
AXL
Lestaurtinib
558
1
AXL
Dactolisib
558
10
AXL
Alpelisib
558
10
AXL
GSK1838705A
558
2
AXL
GSK1838705A
558
2
AXL
PHA-767491
558
3
AXL
BS-181
558
10
AXL
(s)-CR8
558
10
AXL
5z-7-oxozeaenol
558
10
AXL
GW2580
558
10
AXL