Target Affinity Spectrum (TAS) vectors for compounds in the HMS LINCS small molecule library. - Dataset (ID:20000)

The original dataset #20000 (LINCS Compound Protein Targets and Concentrations) with kinase inhibitor target information has been replaced with Target Affinity Spectrum binding information for small molecules in the HMS-LINCS database (March 2019).

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HMSL Small Mol Gene ID Binding Class HUGO Gene Symbol
PP1
558
3
AXL
Sotrastaurin
558
3
AXL
SB202190
558
10
AXL
Axitinib
558
2
AXL
Cediranib
558
2
AXL
Taselisib
558
10
AXL
ABT-737
572
1
BAD
ABT-737
572
1
BAD
Navitoclax
572
1
BAD
Seliciclib
595
10
CCND1
AT-7519
595
2
CCND1
AT-7519
595
2
CCND1
AT-7519
595
2
CCND1
Sorafenib
595
3
CCND1
Sorafenib
595
3
CCND1
Sorafenib
595
3
CCND1
Alvocidib
595
2
CCND1
Alvocidib
595
2
CCND1
Palbociclib
595
1
CCND1
Palbociclib
595
1
CCND1
PHA-793887
595
1
CCND1
Staurosporine
595
1
CCND1
Staurosporine
595
1
CCND1
SNS-032
595
2
CCND1
SNS-032
595
2
CCND1