Small molecules

HMS LINCS ID Name Alternative Names LINCS ID Structure Image PubChem CID
10101-101 PD0325901
PD-325901
LSM-1101 9826528
10464-101 GTPL6019
PDGF receptor tyrosine kinase inhibitor III; 4-(6,7-Dimethoxy-4-quinazolinyl)-N-(4-phenoxyphenyl)-1-piperazinecarboxamide
10907042
10467-101 JNJ-10198409
PDGF receptor tyrosine kinase inhibitor IV
9797370
10222-101 Dacomitinib
PF-00299804
LSM-42808 57519532
10027-101 Crizotinib
PF02341066
LSM-1027 11626560
10027-999 Crizotinib
PF02341066
LSM-1027 11626560
10621-101 Defactinib
PF-04554878; VS-6063
25117126
10243-999 CGC-11047
PG11047
LSM-4266 476863
10047-101 Pictilisib
Pictrelisib; GDC-0941; RG-7321
LSM-1047 17755052
10047-999 Pictilisib
Pictrelisib; GDC-0941; RG-7321
LSM-1047 17755052
10472-101 ST50842732
PIM1/2 Kinase Inhibitor VI
6076476
10119-101 SU11274
PKI-SU11274
LSM-42791 53396327
11951-101 HY-17542
PLpro Inhibitor
44235889
10068-101 Vemurafenib
PLX4032; RG7204; R7204; RO5185426
LSM-1068 42611257
10384-101 SR-2516
PND-1186
25073775
10345-101 Torkinib
PP242
LSM-6357 57347681
10345-111 Torkinib
PP242
LSM-6357 57347681
10345-999 Torkinib
PP242
LSM-6357 57347681
10310-101 Belinostat
PXD101
LSM-43181 53437714
10235-101 Everolimus
RAD001
LSM-4258 53398658
10052-101 Sirolimus
Rapamycin
LSM-1052 5040
10444-101 Cediranib
Recentin; AZD2171
9933475
10418-101 Lenalidomide
Revlimid; CC5013
216326
10234-101 GDC-0980
RG7422
LSM-4257 66694608
10264-999 Methotrexate
Rheumatrex; Trexall; Amethopterin; MTX
LSM-5690 126941