Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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A-375 | Vemurafenib | Trametinib | PF562271 | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 3 | 2640 | 338 | 0.1157 | 0.1234 | 0.1280 | 0.1122 |
WM-115 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2644 | 476 | 0.5083 | 0.5260 | 0.1800 | 0.1772 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2655 | 180 | 0.6416 | 0.6483 | 0.0678 | 0.0808 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 2657 | 368 | 0.1360 | 0.1328 | 0.1385 | 0.1351 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 2 | 2659 | 360 | 0.1366 | 0.1298 | 0.1354 | 0.1284 |
WM-115 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2691 | 483 | 0.5177 | 0.5260 | 0.1795 | 0.1772 |
A-375 | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2696 | 260 | 0.1224 | 0.1221 | 0.0964 | 0.0950 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2715 | 551 | 0.4214 | 0.3998 | 0.2029 | 0.2252 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 2717 | 113 | 0.1673 | 0.1595 | 0.0416 | 0.0410 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 3 | 2720 | 384 | 0.1377 | 0.1271 | 0.1412 | 0.1561 |
WM-115 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 2722 | 220 | 0.6603 | 0.7205 | 0.0808 | 0.0832 |
A-375 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2727 | 252 | 0.1809 | 0.2238 | 0.0924 | 0.0934 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2729 | 242 | 0.6447 | 0.6483 | 0.0887 | 0.0808 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2732 | 645 | 0.4064 | 0.3998 | 0.2361 | 0.2252 |
A-375 | Vemurafenib | Trametinib | Defactinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 2738 | 358 | 0.1347 | 0.1291 | 0.1308 | 0.1308 |
WM-115 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 2739 | 569 | 0.5088 | 0.5131 | 0.2077 | 0.2141 |
WM-115 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 2741 | 592 | 0.5039 | 0.5131 | 0.2160 | 0.2141 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 2 | 2742 | 331 | 0.1421 | 0.1372 | 0.1207 | 0.1215 |
A-375 | Vemurafenib | Trametinib | PF562271 | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 1 | 2750 | 291 | 0.1236 | 0.1234 | 0.1058 | 0.1122 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2752 | 288 | 0.7312 | 0.5728 | 0.1047 | 0.0984 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 2 | 2768 | 450 | 0.1367 | 0.1271 | 0.1626 | 0.1561 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2779 | 239 | 0.6585 | 0.6483 | 0.0860 | 0.0808 |
MZ7-mel | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2786 | 159 | 0.8979 | 0.7564 | 0.0571 | 0.0560 |
A-375 | Vemurafenib | Trametinib | PF562271 | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 1 | 2793 | 297 | 0.1254 | 0.1292 | 0.1063 | 0.1109 |
COLO 858 | Vemurafenib | Trametinib | I-BET151 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2817 | 383 | 0.5973 | 0.4915 | 0.1360 | 0.1414 |