Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2779 | 239 | 0.6585 | 0.6483 | 0.0860 | 0.0808 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2729 | 242 | 0.6447 | 0.6483 | 0.0887 | 0.0808 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2655 | 180 | 0.6416 | 0.6483 | 0.0678 | 0.0808 |
WM-115 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2431 | 184 | 0.6441 | 0.6307 | 0.0757 | 0.0825 |
WM-115 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2490 | 221 | 0.6505 | 0.6307 | 0.0888 | 0.0825 |
WM-115 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2273 | 189 | 0.5974 | 0.6307 | 0.0832 | 0.0825 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 2300 | 197 | 0.6241 | 0.5409 | 0.0857 | 0.0829 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 2464 | 221 | 0.6656 | 0.5409 | 0.0897 | 0.0829 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 1211 | 89 | 0.3330 | 0.5409 | 0.0735 | 0.0829 |
A-375 | Vemurafenib | Trametinib | I-BET151 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 7782 | 655 | 0.4948 | 0.5250 | 0.0842 | 0.0831 |
A-375 | Vemurafenib | Trametinib | I-BET151 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 7321 | 587 | 0.4675 | 0.5250 | 0.0802 | 0.0831 |
A-375 | Vemurafenib | Trametinib | I-BET151 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 9641 | 818 | 0.6126 | 0.5250 | 0.0848 | 0.0831 |
WM-115 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 2722 | 220 | 0.6603 | 0.7205 | 0.0808 | 0.0832 |
WM-115 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 3249 | 292 | 0.7804 | 0.7205 | 0.0899 | 0.0832 |
WM-115 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 2965 | 234 | 0.7208 | 0.7205 | 0.0789 | 0.0832 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 14201 | 1526 | 0.9096 | 1.0000 | 0.1075 | 0.0842 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 16108 | 728 | 1.1037 | 1.0000 | 0.0452 | 0.0842 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 1 | 15279 | 1529 | 0.9867 | 1.0000 | 0.1001 | 0.0842 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2538 | 211 | 0.5691 | 0.5869 | 0.0831 | 0.0856 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2821 | 227 | 0.6344 | 0.5869 | 0.0805 | 0.0856 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2513 | 234 | 0.5573 | 0.5869 | 0.0931 | 0.0856 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 1678 | 145 | 0.1100 | 0.1110 | 0.0864 | 0.0898 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 1704 | 156 | 0.1111 | 0.1110 | 0.0915 | 0.0898 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 1717 | 157 | 0.1119 | 0.1110 | 0.0914 | 0.0898 |
WM-115 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 1951 | 168 | 0.4622 | 0.4571 | 0.0861 | 0.0908 |