Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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A-375 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 7367 | 288 | 0.4205 | 0.4663 | 0.0391 | 0.0378 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1575 | 62 | 1.4609 | 1.3505 | 0.0394 | 0.0426 |
MMAC-SF | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 579 | 23 | 0.5505 | 0.6713 | 0.0397 | 0.0438 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 2009 | 80 | 0.1240 | 0.1595 | 0.0398 | 0.0410 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 18030 | 727 | 1.0201 | 1.0000 | 0.0403 | 0.0484 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 1114 | 46 | 1.0312 | 1.0000 | 0.0413 | 0.0416 |
MMAC-SF | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1256 | 52 | 1.1921 | 1.3614 | 0.0414 | 0.0486 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 628 | 26 | 0.5813 | 0.6350 | 0.0414 | 0.0435 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 3039 | 126 | 0.1872 | 0.1595 | 0.0415 | 0.0410 |
MMAC-SF | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 530 | 22 | 0.5030 | 0.7059 | 0.0415 | 0.0474 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 19598 | 815 | 1.1074 | 1.0240 | 0.0416 | 0.0404 |
A-375 | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 2717 | 113 | 0.1673 | 0.1595 | 0.0416 | 0.0410 |
MZ7-mel | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 3923 | 164 | 0.9907 | 0.9208 | 0.0418 | 0.0457 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 18289 | 776 | 1.0403 | 1.0000 | 0.0424 | 0.0438 |
MMAC-SF | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 872 | 37 | 0.8267 | 0.7521 | 0.0424 | 0.0500 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1538 | 67 | 1.4203 | 1.3505 | 0.0436 | 0.0426 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 16139 | 705 | 0.9168 | 1.0000 | 0.0437 | 0.0438 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 725 | 32 | 0.6691 | 0.6350 | 0.0441 | 0.0435 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 18988 | 841 | 1.0699 | 1.0240 | 0.0443 | 0.0404 |
MMAC-SF | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1712 | 76 | 1.4144 | 1.2637 | 0.0444 | 0.0426 |
A-375 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 2 | 5428 | 243 | 0.3057 | 0.3181 | 0.0448 | 0.0472 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1269 | 57 | 1.1703 | 1.3505 | 0.0449 | 0.0426 |
MZ7-mel | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1710 | 77 | 0.4899 | 0.3534 | 0.0450 | 0.0527 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 710 | 32 | 0.6547 | 0.6350 | 0.0451 | 0.0435 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 16108 | 728 | 1.1037 | 1.0000 | 0.0452 | 0.0842 |