Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
WM-115 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 1 | 2490 | 221 | 0.6505 | 0.6307 | 0.0888 | 0.0825 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2318 | 206 | 0.1255 | 0.1286 | 0.0889 | 0.0918 |
A-375 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 3905 | 348 | 0.2600 | 0.2238 | 0.0891 | 0.0934 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 2464 | 221 | 0.6656 | 0.5409 | 0.0897 | 0.0829 |
WM-115 | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 3249 | 292 | 0.7804 | 0.7205 | 0.0899 | 0.0832 |
A-375 | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 2432 | 219 | 0.1112 | 0.1221 | 0.0900 | 0.0950 |
A-375 | Vemurafenib | Trametinib | I-BET151 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 1694 | 153 | 0.1070 | 0.1100 | 0.0903 | 0.1113 |
WM-115 | Vemurafenib | Trametinib | Belinostat | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 1824 | 165 | 0.4850 | 0.4681 | 0.0905 | 0.0978 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.3160 | 0.0316 | 0.3160 | uM | 72 | hr | 1 | 1508 | 137 | 0.0814 | 0.0866 | 0.0908 | 0.1048 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 1717 | 157 | 0.1119 | 0.1110 | 0.0914 | 0.0898 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 7553 | 690 | 0.4925 | 0.5962 | 0.0914 | 0.0732 |
WM-115 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 3 | 3017 | 276 | 0.6826 | 0.7484 | 0.0915 | 0.0918 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 1704 | 156 | 0.1111 | 0.1110 | 0.0915 | 0.0898 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 2374 | 218 | 0.1281 | 0.1286 | 0.0918 | 0.0918 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2177 | 201 | 0.5864 | 0.5728 | 0.0923 | 0.0984 |
A-375 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 3 | 2727 | 252 | 0.1809 | 0.2238 | 0.0924 | 0.0934 |
A-375 | Vemurafenib | Trametinib | Belinostat | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 2 | 1537 | 143 | 0.1054 | 0.1039 | 0.0930 | 0.1135 |
WM-115 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 2513 | 234 | 0.5573 | 0.5869 | 0.0931 | 0.0856 |
A-375 | Vemurafenib | Trametinib | Belinostat | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 2 | 1755 | 165 | 0.1202 | 0.1127 | 0.0940 | 0.1173 |
A-375 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 1.0000 | uM | 72 | hr | 2 | 9244 | 871 | 0.6009 | 0.5962 | 0.0942 | 0.0732 |
A-375 | Vemurafenib | Trametinib | Saracatinib | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 3 | 2461 | 233 | 0.1323 | 0.1286 | 0.0947 | 0.0918 |
A-375 | Vemurafenib | Trametinib | Belinostat | 0.3160 | 0.0316 | 0.0000 | uM | 72 | hr | 1 | 1507 | 144 | 0.1031 | 0.1039 | 0.0956 | 0.1135 |
A-375 | Vemurafenib | Trametinib | (+)-JQ1 | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 2 | 1660 | 159 | 0.1097 | 0.1126 | 0.0958 | 0.0954 |
A-375 | Vemurafenib | Trametinib | (+)-JQ1 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 2 | 1574 | 151 | 0.1040 | 0.1029 | 0.0959 | 0.1185 |
A-375 | Vemurafenib | Trametinib | PF562271 | 0.1000 | 0.0100 | 0.0000 | uM | 72 | hr | 1 | 2696 | 260 | 0.1224 | 0.1221 | 0.0964 | 0.0950 |