Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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MZ7-mel | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 4494 | 264 | 1.4458 | 1.4565 | 0.0587 | 0.0668 |
MMAC-SF | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1533 | 83 | 1.4356 | 1.3614 | 0.0541 | 0.0486 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 5152 | 346 | 1.4263 | 1.4011 | 0.0672 | 0.0616 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1538 | 67 | 1.4203 | 1.3505 | 0.0436 | 0.0426 |
MMAC-SF | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1585 | 85 | 1.4191 | 1.3504 | 0.0536 | 0.0554 |
MMAC-SF | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1712 | 76 | 1.4144 | 1.2637 | 0.0444 | 0.0426 |
MMAC-SF | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1446 | 46 | 1.3861 | 1.3106 | 0.0318 | 0.0383 |
MMAC-SF | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 1681 | 85 | 1.3798 | 1.2637 | 0.0506 | 0.0426 |
MZ7-mel | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 3.1600 | uM | 72 | hr | 1 | 5474 | 256 | 1.3752 | 0.9655 | 0.0468 | 0.0440 |
MMAC-SF | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1474 | 69 | 1.3292 | 1.3504 | 0.0468 | 0.0554 |
MZ7-mel | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 5776 | 371 | 1.3291 | 1.2673 | 0.0642 | 0.0549 |
MMAC-SF | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 1390 | 63 | 1.3139 | 1.3106 | 0.0453 | 0.0383 |
MMAC-SF | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1474 | 97 | 1.3027 | 1.3504 | 0.0658 | 0.0554 |
MZ7-mel | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 2 | 5542 | 297 | 1.2898 | 1.2673 | 0.0536 | 0.0549 |
MMAC-SF | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1293 | 49 | 1.2317 | 1.3106 | 0.0379 | 0.0383 |
MMAC-SF | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1256 | 52 | 1.1921 | 1.3614 | 0.0414 | 0.0486 |
COLO 858 | Vemurafenib | Trametinib | Belinostat | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 6638 | 1181 | 1.1834 | 1.0000 | 0.1779 | 0.1777 |
MZ7-mel | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 5047 | 236 | 1.1830 | 1.2673 | 0.0468 | 0.0549 |
COLO 858 | Vemurafenib | Trametinib | (+)-JQ1 | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 5108 | 970 | 1.1788 | 1.0000 | 0.1899 | 0.1930 |
MMAC-SF | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 1269 | 57 | 1.1703 | 1.3505 | 0.0449 | 0.0426 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 7119 | 1168 | 1.1589 | 0.9999 | 0.1641 | 0.1645 |
COLO 858 | Vemurafenib | Trametinib | I-BET | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 4941 | 870 | 1.1528 | 1.0000 | 0.1761 | 0.1901 |
MMAC-SF | Vemurafenib | Trametinib | Dasatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 1301 | 83 | 1.1523 | 1.0000 | 0.0638 | 0.0561 |
MMAC-SF | Vemurafenib | Trametinib | Saracatinib | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 1203 | 41 | 1.1505 | 1.0000 | 0.0341 | 0.0425 |
COLO 858 | Vemurafenib | Trametinib | I-BET151 | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 5057 | 491 | 1.1205 | 1.0000 | 0.0971 | 0.0991 |