Viability and apoptosis measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of three compounds (viability/apoptosis dataset 2 of 2) - Dataset (ID:20273)
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Cell | Small Molecule 1 | Small Molecule 2 | Small Molecule 3 | Small Mol 1 Concentration | Small Mol 2 Concentration | Small Mol 3 Concentration | Small Mol Conc Unit | Time Point | Time Point Unit | Replicate | Total Number of Cells (Nuclei) | Number of Apoptotic Cells | Relative Viability | Mean Relative Viability | Apoptosis Fraction | Mean Apoptosis Fraction |
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COLO 858 | Vemurafenib | Trametinib | (+)-JQ1 | 0.1000 | 0.0100 | 1.0000 | uM | 72 | hr | 1 | 1324 | 1269 | 0.0157 | 0.0146 | 0.9585 | 0.9538 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 3 | 1598 | 1262 | 0.0473 | 0.0435 | 0.7897 | 0.7870 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 3 | 1579 | 1242 | 0.0509 | 0.0532 | 0.7866 | 0.7386 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 1402 | 1236 | 0.0251 | 0.0186 | 0.8816 | 0.9092 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 3.1600 | 0.3160 | 1.0000 | uM | 72 | hr | 1 | 1274 | 1219 | 0.0107 | 0.0091 | 0.9568 | 0.9558 |
COLO 858 | Vemurafenib | Trametinib | Dasatinib | 0.1000 | 0.0100 | 3.1600 | uM | 72 | hr | 1 | 1337 | 1219 | 0.0196 | 0.0145 | 0.9117 | 0.9231 |
COLO 858 | Vemurafenib | Trametinib | Dasatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 3 | 1524 | 1214 | 0.0514 | 0.0529 | 0.7966 | 0.7685 |
A-375 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 21851 | 1210 | 1.0372 | 1.0000 | 0.0554 | 0.0502 |
COLO 858 | Vemurafenib | Trametinib | Dasatinib | 3.1600 | 0.3160 | 1.0000 | uM | 72 | hr | 2 | 1237 | 1209 | 0.0046 | 0.0049 | 0.9774 | 0.9743 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 3.1600 | 0.3160 | 1.0000 | uM | 72 | hr | 1 | 1491 | 1204 | 0.0433 | 0.0226 | 0.8075 | 0.8932 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 1 | 1330 | 1201 | 0.0182 | 0.0136 | 0.9030 | 0.9358 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 3.1600 | 0.3160 | 1.0000 | uM | 72 | hr | 2 | 1240 | 1189 | 0.0072 | 0.0087 | 0.9589 | 0.9527 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 2 | 8288 | 1188 | 1.0719 | 1.0000 | 0.1433 | 0.1414 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 1.0000 | 0.1000 | 1.0000 | uM | 72 | hr | 1 | 1403 | 1186 | 0.0328 | 0.0286 | 0.8453 | 0.8489 |
COLO 858 | Vemurafenib | Trametinib | Belinostat | 0.0000 | 0.0000 | 0.0000 | uM | 72 | hr | 3 | 6638 | 1181 | 1.1834 | 1.0000 | 0.1779 | 0.1777 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 2 | 1509 | 1177 | 0.0467 | 0.0435 | 0.7800 | 0.7870 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 0.3160 | 0.0316 | 3.1600 | uM | 72 | hr | 1 | 1324 | 1177 | 0.0222 | 0.0219 | 0.8890 | 0.8885 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 1238 | 1176 | 0.0121 | 0.0135 | 0.9499 | 0.9372 |
COLO 858 | Vemurafenib | Trametinib | Dasatinib | 0.1000 | 0.0100 | 0.3160 | uM | 72 | hr | 3 | 1204 | 1175 | 0.0048 | 0.0045 | 0.9759 | 0.9731 |
COLO 858 | Vemurafenib | Trametinib | PF562271 | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 3 | 7119 | 1168 | 1.1589 | 0.9999 | 0.1641 | 0.1645 |
COLO 858 | Vemurafenib | Trametinib | Defactinib | 0.0000 | 0.0000 | 0.3160 | uM | 72 | hr | 1 | 7512 | 1166 | 0.8932 | 0.9286 | 0.1552 | 0.1630 |
WM-115 | Vemurafenib | Trametinib | JNK-IN-8 | 1.0000 | 0.1000 | 3.1600 | uM | 72 | hr | 2 | 1738 | 1161 | 0.1437 | 0.1262 | 0.6680 | 0.6643 |
COLO 858 | Vemurafenib | Trametinib | JNK-IN-8 | 0.3160 | 0.0316 | 3.1600 | uM | 72 | hr | 3 | 1291 | 1160 | 0.0198 | 0.0219 | 0.8985 | 0.8885 |
COLO 858 | Vemurafenib | Trametinib | Saracatinib | 1.0000 | 0.1000 | 0.0000 | uM | 72 | hr | 3 | 1461 | 1159 | 0.0506 | 0.0484 | 0.7933 | 0.7812 |
MZ7-mel | Vemurafenib | Trametinib | Defactinib | 3.1600 | 0.3160 | 0.0000 | uM | 72 | hr | 3 | 2097 | 1153 | 0.2801 | 0.2264 | 0.5498 | 0.5573 |