Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib AKT2 93.0 100
nM
Taselisib AKT2 99.0 1000
nM
Taselisib AKT3 97.0 100
nM
Taselisib AKT3 95.0 1000
nM
Taselisib ALK 86.0 100
nM
Taselisib ALK 100.0 1000
nM
Taselisib ALK(C1156Y) 79.0 100
nM
Taselisib ALK(C1156Y) 87.0 1000
nM
Taselisib ALK(L1196M) 78.0 100
nM
Taselisib ALK(L1196M) 74.0 1000
nM
Taselisib AMPK-alpha1 93.0 100
nM
Taselisib AMPK-alpha1 90.0 1000
nM
Taselisib AMPK-alpha2 89.0 100
nM
Taselisib AMPK-alpha2 99.0 1000
nM
Taselisib ANKK1 90.0 100
nM
Taselisib ANKK1 89.0 1000
nM
Taselisib NUAK1 97.0 100
nM
Taselisib NUAK1 100.0 1000
nM
Taselisib M3K5 97.0 100
nM
Taselisib M3K5 100.0 1000
nM
Taselisib M3K6 77.0 100
nM
Taselisib M3K6 88.0 1000
nM
Taselisib AURKA 97.0 100
nM
Taselisib AURKA 100.0 1000
nM
Taselisib AURKB 91.0 100
nM