BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | PIK4CB | 7.7 | 1000 | nM |
Alpelisib | FYV1 | 93.0 | 100 | nM |
Alpelisib | FYV1 | 98.0 | 1000 | nM |
Alpelisib | PIM1 | 87.0 | 100 | nM |
Alpelisib | PIM1 | 100.0 | 1000 | nM |
Alpelisib | PIM2 | 85.0 | 100 | nM |
Alpelisib | PIM2 | 100.0 | 1000 | nM |
Alpelisib | PIM3 | 79.0 | 100 | nM |
Alpelisib | PIM3 | 93.0 | 1000 | nM |
Alpelisib | PIP5K1A | 92.0 | 100 | nM |
Alpelisib | PIP5K1A | 100.0 | 1000 | nM |
Alpelisib | PIP5K1C | 86.0 | 100 | nM |
Alpelisib | PIP5K1C | 83.0 | 1000 | nM |
Alpelisib | PIP5K2B | 100.0 | 100 | nM |
Alpelisib | PIP5K2B | 76.0 | 1000 | nM |
Alpelisib | PI42C | 100.0 | 100 | nM |
Alpelisib | PI42C | 84.0 | 1000 | nM |
Alpelisib | PKAC-alpha | 81.0 | 100 | nM |
Alpelisib | PKAC-alpha | 90.0 | 1000 | nM |
Alpelisib | PKAC-beta | 94.0 | 100 | nM |
Alpelisib | PKAC-beta | 90.0 | 1000 | nM |
Alpelisib | PKMYT1 | 100.0 | 100 | nM |
Alpelisib | PKMYT1 | 90.0 | 1000 | nM |
Alpelisib | PKN1 | 100.0 | 100 | nM |
Alpelisib | PKN1 | 93.0 | 1000 | nM |