BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib PIK4CB 7.7 1000
nM
Alpelisib FYV1 93.0 100
nM
Alpelisib FYV1 98.0 1000
nM
Alpelisib PIM1 87.0 100
nM
Alpelisib PIM1 100.0 1000
nM
Alpelisib PIM2 85.0 100
nM
Alpelisib PIM2 100.0 1000
nM
Alpelisib PIM3 79.0 100
nM
Alpelisib PIM3 93.0 1000
nM
Alpelisib PIP5K1A 92.0 100
nM
Alpelisib PIP5K1A 100.0 1000
nM
Alpelisib PIP5K1C 86.0 100
nM
Alpelisib PIP5K1C 83.0 1000
nM
Alpelisib PIP5K2B 100.0 100
nM
Alpelisib PIP5K2B 76.0 1000
nM
Alpelisib PI42C 100.0 100
nM
Alpelisib PI42C 84.0 1000
nM
Alpelisib PKAC-alpha 81.0 100
nM
Alpelisib PKAC-alpha 90.0 1000
nM
Alpelisib PKAC-beta 94.0 100
nM
Alpelisib PKAC-beta 90.0 1000
nM
Alpelisib PKMYT1 100.0 100
nM
Alpelisib PKMYT1 90.0 1000
nM
Alpelisib PKN1 100.0 100
nM
Alpelisib PKN1 93.0 1000
nM