BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib MAP3K4 100.0 100
nM
Alpelisib MAP3K4 100.0 1000
nM
Alpelisib MAP4K2 100.0 100
nM
Alpelisib MAP4K2 100.0 1000
nM
Alpelisib MAP4K4 100.0 1000
nM
Alpelisib MAP4K4 94.0 100
nM
Alpelisib MAP4K5 94.0 1000
nM
Alpelisib MAP4K5 91.0 100
nM
Alpelisib MAPKAPK2 100.0 1000
nM
Alpelisib MAPKAPK2 100.0 100
nM
Alpelisib MAPKAPK5 100.0 1000
nM
Alpelisib MAPKAPK5 100.0 100
nM
Alpelisib MARK1 100.0 100
nM
Alpelisib MARK1 92.0 1000
nM
Alpelisib MARK2 100.0 100
nM
Alpelisib MARK2 100.0 1000
nM
Alpelisib MARK3 100.0 100
nM
Alpelisib MARK3 100.0 1000
nM
Alpelisib MARK4 95.0 1000
nM
Alpelisib MARK4 100.0 100
nM
Alpelisib MAST1 100.0 1000
nM
Alpelisib MAST1 100.0 100
nM
Alpelisib MELK 86.0 1000
nM
Alpelisib MELK 91.0 100
nM
Alpelisib MERTK 100.0 100
nM