BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | EPHB4 | 81.0 | 100 | nM |
Alpelisib | EPHB6 | 100.0 | 1000 | nM |
Alpelisib | EPHB6 | 100.0 | 100 | nM |
Alpelisib | ERBB2 | 89.0 | 100 | nM |
Alpelisib | ERBB2 | 89.0 | 1000 | nM |
Alpelisib | ERBB3 | 100.0 | 1000 | nM |
Alpelisib | ERBB3 | 100.0 | 100 | nM |
Alpelisib | ERBB4 | 100.0 | 1000 | nM |
Alpelisib | ERBB4 | 100.0 | 100 | nM |
Alpelisib | ERK3 | 100.0 | 100 | nM |
Alpelisib | ERK3 | 100.0 | 1000 | nM |
Alpelisib | ERK4 | 100.0 | 1000 | nM |
Alpelisib | ERK4 | 97.0 | 100 | nM |
Alpelisib | ERK5 | 97.0 | 100 | nM |
Alpelisib | ERK5 | 100.0 | 1000 | nM |
Alpelisib | ERK8 | 100.0 | 100 | nM |
Alpelisib | ERK8 | 100.0 | 1000 | nM |
Alpelisib | ERN1 | 100.0 | 1000 | nM |
Alpelisib | ERN1 | 100.0 | 100 | nM |
Alpelisib | FAK1 | 100.0 | 1000 | nM |
Alpelisib | FAK1 | 84.0 | 100 | nM |
Alpelisib | FAK2 | 100.0 | 1000 | nM |
Alpelisib | FAK2 | 99.0 | 100 | nM |
Alpelisib | FER | 92.0 | 1000 | nM |
Alpelisib | FER | 74.0 | 100 | nM |