BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib DYRK2 94.0 100
nM
Alpelisib EGFR 100.0 1000
nM
Alpelisib EGFR 97.0 100
nM
Alpelisib EGFR(E746-A750del) 93.0 1000
nM
Alpelisib EGFR(E746-A750del) 100.0 100
nM
Alpelisib EGFR(G719C) 100.0 100
nM
Alpelisib EGFR(G719C) 100.0 1000
nM
Alpelisib EGFR(G719S) 96.0 1000
nM
Alpelisib EGFR(G719S) 100.0 100
nM
Alpelisib EGFR(L747-E749del, A750P) 97.0 1000
nM
Alpelisib EGFR(L747-E749del, A750P) 99.0 100
nM
Alpelisib EGFR(L747-S752del, P753S) 92.0 1000
nM
Alpelisib EGFR(L747-S752del, P753S) 96.0 100
nM
Alpelisib EGFR(L747-T751del,Sins) 96.0 100
nM
Alpelisib EGFR(L747-T751del,Sins) 78.0 1000
nM
Alpelisib EGFR(L858R) 95.0 100
nM
Alpelisib EGFR(L858R) 100.0 1000
nM
Alpelisib EGFR(L858R,T790M) 100.0 1000
nM
Alpelisib EGFR(L858R,T790M) 94.0 100
nM
Alpelisib EGFR(L861Q) 82.0 1000
nM
Alpelisib EGFR(L861Q) 96.0 100
nM
Alpelisib EGFR(S752-I759del) 100.0 100
nM
Alpelisib EGFR(S752-I759del) 98.0 1000
nM
Alpelisib EGFR(T790M) 100.0 100
nM
Alpelisib EGFR(T790M) 100.0 1000
nM