BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib PAK4 65.0 100
nM
Alpelisib TNK1 67.0 1000
nM
Alpelisib CSF1R-autoinhibited 67.0 100
nM
Alpelisib SLK 69.0 100
nM
Alpelisib CAMK1 69.0 100
nM
Alpelisib CLK4 69.0 100
nM
Alpelisib PAK2 69.0 100
nM
Alpelisib PIK3CD 70.0 100
nM
Alpelisib CASK 71.0 1000
nM
Alpelisib DRAK1 72.0 1000
nM
Alpelisib RSK2(Kin.Dom.2-C-terminal) 72.0 100
nM
Alpelisib IRAK3 72.0 1000
nM
Alpelisib MLK3 73.0 100
nM
Alpelisib CAMK1D 73.0 100
nM
Alpelisib HIPK4 73.0 100
nM
Alpelisib ABL1(F317I)-phosphorylated 73.0 1000
nM
Alpelisib MP2K2 74.0 100
nM
Alpelisib ABL1(Q252H)-nonphosphorylated 74.0 1000
nM
Alpelisib FER 74.0 100
nM
Alpelisib TLK2 74.0 100
nM
Alpelisib PAK1 75.0 100
nM
Alpelisib AAK1 75.0 1000
nM
Alpelisib TLK1 76.0 1000
nM
Alpelisib RSK4(Kin.Dom.2-C-terminal) 76.0 100
nM
Alpelisib PIP5K2B 76.0 1000
nM