BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | PAK4 | 65.0 | 100 | nM |
Alpelisib | TNK1 | 67.0 | 1000 | nM |
Alpelisib | CSF1R-autoinhibited | 67.0 | 100 | nM |
Alpelisib | SLK | 69.0 | 100 | nM |
Alpelisib | CAMK1 | 69.0 | 100 | nM |
Alpelisib | CLK4 | 69.0 | 100 | nM |
Alpelisib | PAK2 | 69.0 | 100 | nM |
Alpelisib | PIK3CD | 70.0 | 100 | nM |
Alpelisib | CASK | 71.0 | 1000 | nM |
Alpelisib | DRAK1 | 72.0 | 1000 | nM |
Alpelisib | RSK2(Kin.Dom.2-C-terminal) | 72.0 | 100 | nM |
Alpelisib | IRAK3 | 72.0 | 1000 | nM |
Alpelisib | MLK3 | 73.0 | 100 | nM |
Alpelisib | CAMK1D | 73.0 | 100 | nM |
Alpelisib | HIPK4 | 73.0 | 100 | nM |
Alpelisib | ABL1(F317I)-phosphorylated | 73.0 | 1000 | nM |
Alpelisib | MP2K2 | 74.0 | 100 | nM |
Alpelisib | ABL1(Q252H)-nonphosphorylated | 74.0 | 1000 | nM |
Alpelisib | FER | 74.0 | 100 | nM |
Alpelisib | TLK2 | 74.0 | 100 | nM |
Alpelisib | PAK1 | 75.0 | 100 | nM |
Alpelisib | AAK1 | 75.0 | 1000 | nM |
Alpelisib | TLK1 | 76.0 | 1000 | nM |
Alpelisib | RSK4(Kin.Dom.2-C-terminal) | 76.0 | 100 | nM |
Alpelisib | PIP5K2B | 76.0 | 1000 | nM |