BYL719 KINOMEscan - Dataset (ID:20263)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | PIK3CA(H1047Y) | 15.0 | 1000 | nM |
Alpelisib | ABL1(H396P)-nonphosphorylated | 16.0 | 1000 | nM |
Alpelisib | PIK3CD | 20.0 | 1000 | nM |
Alpelisib | PHKG1 | 20.0 | 1000 | nM |
Alpelisib | HIPK4 | 39.0 | 1000 | nM |
Alpelisib | ABL1(F317I)-nonphosphorylated | 44.0 | 1000 | nM |
Alpelisib | DYRK1B | 45.0 | 1000 | nM |
Alpelisib | CLK2 | 45.0 | 1000 | nM |
Alpelisib | PIK3C2G | 50.0 | 1000 | nM |
Alpelisib | ABL1-nonphosphorylated | 53.0 | 1000 | nM |
Alpelisib | ABL1(F317L)-phosphorylated | 53.0 | 1000 | nM |
Alpelisib | DYRK1B | 54.0 | 100 | nM |
Alpelisib | SYK | 58.0 | 100 | nM |
Alpelisib | MYLK | 59.0 | 100 | nM |
Alpelisib | CLK4 | 59.0 | 1000 | nM |
Alpelisib | CLK1 | 59.0 | 1000 | nM |
Alpelisib | RSK4(Kin.Dom.2-C-terminal) | 61.0 | 1000 | nM |
Alpelisib | MTOR | 61.0 | 1000 | nM |
Alpelisib | ABL1(H396P)-nonphosphorylated | 63.0 | 100 | nM |
Alpelisib | RIOK1 | 64.0 | 100 | nM |
Alpelisib | LCK | 65.0 | 100 | nM |
Alpelisib | NEK5 | 65.0 | 100 | nM |
Alpelisib | ABL1(F317L)-nonphosphorylated | 65.0 | 1000 | nM |
Alpelisib | CDKL1 | 65.0 | 100 | nM |
Alpelisib | PAK4 | 65.0 | 100 | nM |