BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib PIK3CA(H1047Y) 15.0 1000
nM
Alpelisib ABL1(H396P)-nonphosphorylated 16.0 1000
nM
Alpelisib PIK3CD 20.0 1000
nM
Alpelisib PHKG1 20.0 1000
nM
Alpelisib HIPK4 39.0 1000
nM
Alpelisib ABL1(F317I)-nonphosphorylated 44.0 1000
nM
Alpelisib DYRK1B 45.0 1000
nM
Alpelisib CLK2 45.0 1000
nM
Alpelisib PIK3C2G 50.0 1000
nM
Alpelisib ABL1-nonphosphorylated 53.0 1000
nM
Alpelisib ABL1(F317L)-phosphorylated 53.0 1000
nM
Alpelisib DYRK1B 54.0 100
nM
Alpelisib SYK 58.0 100
nM
Alpelisib MYLK 59.0 100
nM
Alpelisib CLK4 59.0 1000
nM
Alpelisib CLK1 59.0 1000
nM
Alpelisib RSK4(Kin.Dom.2-C-terminal) 61.0 1000
nM
Alpelisib MTOR 61.0 1000
nM
Alpelisib ABL1(H396P)-nonphosphorylated 63.0 100
nM
Alpelisib RIOK1 64.0 100
nM
Alpelisib LCK 65.0 100
nM
Alpelisib NEK5 65.0 100
nM
Alpelisib ABL1(F317L)-nonphosphorylated 65.0 1000
nM
Alpelisib CDKL1 65.0 100
nM
Alpelisib PAK4 65.0 100
nM